SCHEMBL16004164

SCHEMBL16004164

O=S(=O)(c1ccc(F)c(Cl)c1)N1CCOc2ccc(COCc3ccccc3F)cc2C1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.44
PKM P14618 12/20 0.43
PKLR P30613 10/20 0.43
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
THRB P10828 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
LMNA P02545 2/20 0.39
MAPT P10636 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004325 0.92 RORC (0.44) RORCPKMPKLRNPC1RAB9A
SCHEMBL16004227 0.91 PKM (0.43) RORCPKMPKLRNPC1RAB9A
SCHEMBL16004228 0.90 PKM (0.52) PKMPKLRNPC1RAB9AKDM4E
SCHEMBL16004107 0.86 PKM (0.45) RORCPKMPKLRKDM4ELMNA
SCHEMBL16004163 0.85 PKM (0.49) RORCPKMPKLRNPC1RAB9A
SCHEMBL16004015 0.84 RORC (0.42) RORCPKMPKLRKDM4ELMNA
SCHEMBL16004229 0.84 PKM (0.46) RORCPKMPKLRKDM4ELMNA
SCHEMBL16004262 0.84 L3MBTL1 (0.45) RORCNPC1RAB9AKDM4EPOLB
SCHEMBL16004330 0.81 PKM (0.46) RORCPKMPKLRLMNAALDH1A1
SCHEMBL16004017 0.80 PKM (0.44) RORCPKMPKLRPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed