SCHEMBL16004163

SCHEMBL16004163

COc1cccc(S(=O)(=O)N2CCOc3ccc(COCc4ccccc4F)cc3C2)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 9/20 0.49
PKLR P30613 5/20 0.49
POLB P06746 3/20 0.48
LMNA P02545 2/20 0.46
TSHR P16473 2/20 0.46
MAPK1 P28482 1/20 0.46
RORC P51449 1/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 4/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
AKR1C3 P42330 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004099 0.90 PKM (0.52) PKMPKLRPOLBLMNATSHR
SCHEMBL16004336 0.89 PKM (0.52) PKMPKLRPOLBLMNATSHR
SCHEMBL16004228 0.87 PKM (0.52) PKMPKLRLMNAKDM4EGAA
SCHEMBL16004227 0.86 PKM (0.43) PKMPKLRLMNARORCMAPT
SCHEMBL16004164 0.85 RORC (0.44) PKMPKLRPOLBLMNATSHR
SCHEMBL16004020 0.81 PKM (0.40) PKMPKLRPOLBLMNAMAPT
SCHEMBL16004338 0.81 LMNA (0.39) PKMPKLRLMNAMAPK1RORC
SCHEMBL16004262 0.79 L3MBTL1 (0.45) POLBLMNATSHRMAPK1RORC
SCHEMBL16004230 0.78 PKM (0.46) PKMPKLRLMNAMAPK1RORC
SCHEMBL16004229 0.78 PKM (0.46) PKMPKLRLMNATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed