SCHEMBL16004228

SCHEMBL16004228

O=S(=O)(c1ccc2c(c1)OCCO2)N1CCOc2ccc(COCc3ccccc3F)cc2C1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PKM P14618 19/20 0.52
PKLR P30613 15/20 0.52
LMNA P02545 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16004164 0.90 RORC (0.44) PKMPKLRLMNANPC1RAB9A
SCHEMBL16004010 0.89 PKM (0.55) PKMPKLRLMNANPC1RAB9A
SCHEMBL16004163 0.87 PKM (0.49) PKMPKLRLMNANPC1RAB9A
SCHEMBL16004227 0.87 PKM (0.43) PKMPKLRLMNANPC1RAB9A
SCHEMBL16004107 0.83 PKM (0.45) PKMPKLRLMNAKDM4ESMN1; SMN2
SCHEMBL16004338 0.82 LMNA (0.39) PKMPKLRLMNASMN1; SMN2
SCHEMBL16004020 0.82 PKM (0.40) PKMPKLRLMNARAB9AKDM4E
SCHEMBL16004262 0.82 L3MBTL1 (0.45) LMNANPC1RAB9AKDM4EGAA
SCHEMBL16004006 0.82 GPR142 (0.45) PKMPKLRLMNANPC1RAB9A
SCHEMBL16004325 0.82 RORC (0.44) PKMPKLRLMNANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed