Bromide

Bromide

SCHEMBL160231

Br.BrCc1cccc(P(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
TSHR P16473 2/20 0.50
TRPA1 O75762 1/20 0.50
TDP1 Q9NUW8 2/20 0.48
CYP3A4 P08684 1/20 0.48
ESR1 P03372 2/20 0.39
ESR2 Q92731 2/20 0.39
LOXL2 Q9Y4K0 1/20 0.34
CES2 O00748 2/20 0.33
CES1 P23141 2/20 0.33
CALM1 P0DP23 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
OPRK1 P41145 3/20 0.32
OPRM1 P35372 2/20 0.32
OPRD1 P41143 2/20 0.32
MAOB P27338 3/20 0.31
MAOA P21397 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19678032 0.98 ALDH1A1 (0.52) ALDH1A1TSHRTRPA1TDP1CYP3A4
Benzyl Bromide SCHEMBL1043932 0.85 TSHR (0.70) ALDH1A1TSHRTRPA1TDP1CYP3A4
SCHEMBL4410065 0.85 TRPA1 (0.46) ALDH1A1TSHRTRPA1TDP1CYP3A4
SCHEMBL2646995 0.83 ALDH1A1 (0.45) ALDH1A1TSHRTRPA1TDP1CYP3A4
SCHEMBL5972931 0.83 TRPA1 (0.45) ALDH1A1TSHRTRPA1TDP1CYP3A4
Bromide SCHEMBL5007355 0.82 MAOA (0.50) ALDH1A1TDP1CYP3A4ESR1ESR2
SCHEMBL10982048 0.79 CYP3A4 (0.52) TDP1CYP3A4ESR1ESR2LOXL2
SCHEMBL2647549 0.79 MEN1 (0.52) ALDH1A1TSHRTRPA1CYP3A4CYP1A2
SCHEMBL10584452 0.79 MEP1A (0.43) ALDH1A1TSHRTRPA1TDP1CYP3A4
SCHEMBL5398999 0.79 CALM1 (0.51) TSHRCALM1CYP1A2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140249102-A1 Topical Applicator Composition and Process for Treatment of Radiologically Contaminated Dermal Injuries BATTELLE MEMORIAL INSTITUTE (US) 2014-09-04 US disclosed
WO-2012030429-A1 TOPICAL APPLICATOR COMPOSITION AND PROCESS FOR REMOVAL OF RADIONUCLIDES FROM RADIOLOGICALLY CONTAMINATED DERMAL SURFACES BATTELLE MEMORIAL INSTITUTE (US) 2012-03-08 WO disclosed