SCHEMBL16048828

SCHEMBL16048828

CCCC(O)C(C)C(O)CCC.O=S(=O)(O)c1ccccc1.O=S(=O)(O)c1ccccc1

nearest known ligand 0.53

Known targets — ChEMBL curated mechanism

BTKCACNA1CCACNA1DCACNA1FCACNA1SCACNA2D1CACNA2D2DRD2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQHRH1HTR2AP2RY12

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
PSIP1 O75475 1/20 0.41
POLB P06746 2/20 0.40
CYP2D6 P10635 1/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MMP1 P03956 3/20 0.38
MMP7 P09237 3/20 0.38
MMP12 P39900 3/20 0.38
MMP13 P45452 3/20 0.38
ACE P12821 2/20 0.38
HSD11B1 P28845 1/20 0.38
ALDH1A1 P00352 3/20 0.37
NT5E P21589 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16046060 0.95 TSHR (0.48) TSHRSMN1; SMN2PSIP1POLBCYP2D6
Benzoic Acid SCHEMBL16046814 0.91 SMN1; SMN2 (0.44) TSHRSMN1; SMN2NPC1RAB9AMMP1
Benzoic Acid SCHEMBL16046263 0.88 SMN1; SMN2 (0.41) TSHRSMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL16045650 0.86 TSHR (0.57) TSHRSMN1; SMN2PSIP1POLBCYP2D6
SCHEMBL11359221 0.84 SMN1; SMN2 (0.59) TSHRSMN1; SMN2PSIP1POLBCYP2D6
SCHEMBL28053070 0.83 LMNA (0.48) TSHRSMN1; SMN2POLBCYP2D6NPC1
Ethohexadiol SCHEMBL16046315 0.81 LMNA (0.56) TSHRSMN1; SMN2PSIP1POLBCYP2D6
SCHEMBL16045028 0.81 SMN1; SMN2 (0.55) TSHRSMN1; SMN2PSIP1POLBCYP2D6
SCHEMBL16044868 0.80 TSHR (0.64) TSHRSMN1; SMN2PSIP1POLBCYP2D6
Isopropyl Alcohol SCHEMBL5735328 0.80 TSHR (0.76) TSHRSMN1; SMN2PSIP1POLBCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2969201-B1 NON-PHTHALATE COMPOUNDS AS ELECTRON DONORS FOR POLYOLEFIN CATALYSTS FORMOSA PLASTICS CORP USA (US) 2022-05-04 EP disclosed
US-9790291-B2 Non-phthalate compounds as electron donors for polyolefin catalysts FORMOSA PLASTICS CORPORATION, USA (US) 2017-10-17 US disclosed
EP-2969201-A2 NON-PHTHALATE COMPOUNDS AS ELECTRON DONORS FOR POLYOLEFIN CATALYSTS Formosa Plastics Corporation, U.S.A. (US) 2016-01-20 EP disclosed
WO-2014160012-A2 NON-PHTHALATE COMPOUNDS AS ELECTRON DONORS FOR POLYOLEFIN CATALYSTS FORMOSA PLASTICS CORPORATION, USA (US) 2014-10-02 WO disclosed
US-20140275456-A1 NON-PHTHALATE COMPOUNDS AS ELECTRON DONORS FOR POLYOLEFIN CATALYSTS FORMOSA PLASTICS CORPORATION, USA (US) 2014-09-18 US disclosed