SCHEMBL16062155

SCHEMBL16062155

CC(O)OC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
ALOX15 P16050 1/20 0.41
CYP2D6 P10635 2/20 0.39
CYP1A2 P05177 1/20 0.39
MAPK1 P28482 1/20 0.39
KCNN4 O15554 3/20 0.38
LMNA P02545 2/20 0.38
KIF11 P52732 1/20 0.38
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37
GRIN1 Q05586 4/20 0.36
GRIN2A Q12879 4/20 0.36
GRIN2D O15399 3/20 0.36
GRIN2C Q14957 3/20 0.36
GRIN2B Q13224 2/20 0.36
ESR1 P03372 2/20 0.35
ESR2 Q92731 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2C P18825 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5899999 0.83 ALDH1A1 (0.39) ALDH1A1ALOX15CYP2D6CYP1A2MAPK1
SCHEMBL4367368 0.81 MAPK1 (0.42) ALDH1A1ALOX15CYP2D6CYP1A2MAPK1
SCHEMBL663135 0.80 ALDH1A1 (0.45) ALDH1A1ALOX15CYP2D6CYP1A2MAPK1
SCHEMBL27413509 0.77 MAPK1 (0.39) ALDH1A1ALOX15CYP2D6CYP1A2MAPK1
SCHEMBL8813285 0.77 MAPK1 (0.39) ALDH1A1ALOX15CYP2D6CYP1A2MAPK1
SCHEMBL3812105 0.77 CYP1A2 (0.46) ALDH1A1ALOX15CYP2D6CYP1A2KCNN4
SCHEMBL8868519 0.77 CYP1A2 (0.46) ALDH1A1ALOX15CYP2D6CYP1A2KCNN4
SCHEMBL16551069 0.77 LMNA (0.42) ALDH1A1ALOX15CYP2D6MAPK1KCNN4
SCHEMBL3529955 0.77 TRPA1 (0.38) ALDH1A1ALOX15CYP2D6CYP1A2MAPK1
SCHEMBL3529956 0.77 TRPA1 (0.38) ALDH1A1ALOX15CYP2D6CYP1A2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970147-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-1-((1S,4R, 5S)-2-FLUORO-4,5-DIHYDROXY-3-HYDROXYMETHYL-CYCLOPENT-2-ENYL)-1H-PYRIMIDIN-2-ONE Rexahn Pharmaceuticals, Inc. (US) 2016-01-20 EP disclosed
EP-2845587-A2 Melanin production inhibitor Pola Chemical Industries Inc. (JP) 2015-03-11 EP disclosed
WO-2014145807-A1 PROCESS FOR THE PREPARATION OF 4-AMINO-1-((1S,4R, 5S)-2-FLUORO-4,5-DIHYDROXY-3-HYDROXYMETHYL-CYCLOPENT-2-ENYL)-1H-PYRIMIDIN-2-ONE REXAHN PHARMACEUTICALS, INC. (US) 2014-09-18 WO disclosed