SCHEMBL16100563

SCHEMBL16100563

FC(F)(F)c1nc2n(c1Cc1cc(Cl)cc(Cl)c1)CCNC2

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.34
HTR2C P28335 4/20 0.33
HTR2A P28223 3/20 0.33
ADRB2 P07550 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
ADRB1 P08588 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
LIPG Q9Y5X9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5273467 0.70 ADRB1 (0.30) ADRB1
SCHEMBL10095034 0.68 P2RX7 (0.38)
SCHEMBL7197337 0.66 LIPG (0.39) HTR2CHTR2ALIPG
SCHEMBL5935834 0.65
SCHEMBL10095064 0.65 P2RX7 (0.45) HTR2CHTR2AADRB2LIPG
SCHEMBL19005240 0.64
SCHEMBL109562 0.64 P2RX7 (0.47) HTR2CHTR2A
SCHEMBL28378309 0.62
SCHEMBL24176784 0.62 SLC6A2 (0.37)
SCHEMBL29792014 0.62 SLC6A2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970302-A1 S1P AND/OR ATX MODULATING AGENTS Biogen MA Inc. (US) 2016-01-20 EP disclosed
WO-2014152725-A1 S1P AND/OR ATX MODULATING AGENTS BIOGEN IDEC MA INC. (US) 2014-09-25 WO disclosed