SCHEMBL1611013

SCHEMBL1611013

C/C=[C]/c1cccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHAT P28329 1/20 0.43
ALDH1A1 P00352 6/20 0.43
CYP2A6 P11509 4/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
HSD17B10 Q99714 5/20 0.40
TSHR P16473 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
GRM5 P41594 1/20 0.40
SIGMAR1 Q99720 1/20 0.38
CYP1A2 P05177 6/20 0.38
HPGD P15428 3/20 0.38
CYP3A4 P08684 2/20 0.38
KEAP1 Q14145 1/20 0.38
HPRT1 P00492 1/20 0.37
HTT P42858 1/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
ABCB11 O95342 1/20 0.35
NR3C1 P04150 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1612209 0.82 ALDH1A1 (0.38) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL6003188 0.80 CHAT (0.39) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL1611479 0.78 CHAT (0.40) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL6003313 0.75 CA1 (0.40) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL50728 0.75 CA1 (0.40) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL1610598 0.75 CHAT (0.38) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL59702 0.75 CA1 (0.69) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL5865111 0.75 CA1 (0.47) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL1663806 0.75 ALDH1A1 (0.48) CHATALDH1A1CYP2A6CA1CA2
SCHEMBL1141298 0.74 HPRT1 (0.52) CHATALDH1A1CYP2A6CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116535460-A Sulfur-containing peptidomimetic compounds, and preparation method and application thereof 中国人民解放军军事科学院军事医学研究院 2023-08-04 CN claimed
EP-0319986-B1 Anti-plasmin depressant NIPPON SHINYAKU CO LTD (JP) 1997-03-12 EP claimed
CN-116535460-A Sulfur-containing peptidomimetic compounds, and preparation method and application thereof 中国人民解放军军事科学院军事医学研究院 2023-08-04 CN disclosed
US-7943612-B2 Compounds that modulate PPAR activity, their preparation and use HIGH POINT PHARMACEUTICALS, LLC (US) 2011-05-17 US disclosed
US-20110087034-A1 Organic Semiconductor Material SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2011-04-14 US disclosed
EP-2248818-A1 ORGANIC SEMICONDUCTOR MATERIAL Sumitomo Chemical Company, Limited (JP) 2010-11-10 EP disclosed
US-7557127-B2 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2009-07-07 US disclosed
US-20090054464-A1 HDAC INHIBITOR ASTELLAS PHARMA INC. (JP) 2009-02-26 US disclosed
US-20090048257-A1 COMPOUNDS THAT MODULATE PPAR ACTIVITY, THEIR PREPARATION AND USE HIGH POINT PHARMACEUTICALS, LLC 2009-02-19 US disclosed
US-7465731-B2 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2008-12-16 US disclosed
EP-1999098-A2 COMPOUNDS THAT MODULATE PPAR ACTIVITY, THEIR PREPARATION AND USE High Point Pharmaceuticals, LLC (US) 2008-12-10 EP disclosed
EP-0319986-B1 Anti-plasmin depressant NIPPON SHINYAKU CO LTD (JP) 1997-03-12 EP disclosed
US-5292750-A piperidine compounds NIPPON SHINYAKU CO. LTD. (JP) 1994-03-08 US disclosed
US-5192772-A Administering moranoline derivatives; anticoagulants NIPPON SHINYAKU CO. LTD. (JP) 1993-03-09 US disclosed
EP-0498680-A1 New beta-amino-alpha-hydroxycarboxylic acids and their use Sankyo Company Limited (JP) 1992-08-12 EP disclosed
EP-0319986-A2 Fibrinolytic agents NIPPON SHINYAKU COMPANY, LIMITED (JP) 1989-06-14 EP disclosed
US-4576753-A MICROBIOCIDES, ANTIBIOTICS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1986-03-18 US disclosed
US-4304718-A ANTIBIOTICS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-12-08 US disclosed
US-4264498-A REACTED WITH AN ACID, ITS ACID HALIDE, OR ANHYDRIDE IN THE PRESENCE OF BORON TRIHALIDE AND AN ORGANIC BASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-04-28 US disclosed
US-4181800-A ANTIBIOTICS FROM SUBSTITUTED PERHYDRO-S-TRIAZINES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-01-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048257-A1 COMPOUNDS THAT MODULATE PPAR ACTIVITY, THEIR PREPARATION AND USE PPARD, PPARG, PPARA CHAT 2548/4885ALDH1A1 1075/4885CYP2A6 326/4885
US-20090054464-A1 HDAC INHIBITOR HDAC1, HDAC2, HDAC8 CHAT 3056/4885ALDH1A1 739/4885CYP2A6 2233/4885
US-20110087034-A1 Organic Semiconductor Material OR10J3, TST, OR51E2 CHAT 1928/4885ALDH1A1 137/4885CYP2A6 1465/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.