SCHEMBL16166195

SCHEMBL16166195

CC(c1ccc(C(F)(F)F)cc1)n1nnc(C(=O)O)c1N

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 10/20 0.42
PTGDR2 Q9Y5Y4 3/20 0.40
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
PTGER4 P35408 1/20 0.38
PDE9A O76083 1/20 0.38
DPP4 P27487 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
GPR139 Q6DWJ6 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
BRD4 O60885 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16166256 0.83 HPGD (0.43) PTGDR2GPR139GAABRD4HPGD
SCHEMBL25064660 0.81 HPGD (0.44) ALDH1A1HPGD
SCHEMBL12377286 0.74 ALDH1A1 (0.50) DPP4DPP7ALDH1A1GAAHPGD
SCHEMBL18290696 0.71 PDE2A (0.49) PDE2APTGDR2PDE9ABRD4
SCHEMBL18282858 0.71 PDE2A (0.49) PDE2APTGDR2PDE9ABRD4
SCHEMBL11483545 0.70 CES2 (0.46) PDE2APTGDR2CES2CES1PTGER4
SCHEMBL16166240 0.70 PDE2A (0.44) PDE2APDE9A
SCHEMBL20150749 0.68 PDE2A (0.52) PDE2APTGDR2PDE9A
SCHEMBL29092145 0.68 PDE2A (0.44) PDE2APTGDR2PDE9ABRD4
SCHEMBL29092133 0.68 PDE2A (0.44) PDE2APTGDR2PDE9ABRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014167528-A1 SPIROPYRAZOLOPYRIDINE DERIVATIVES AND USES THEREOF FOR THE TREATMENT OF VIRAL INFECTIONS NOVARTIS AG (CH) 2014-10-16 WO disclosed
WO-2014167528-A1 SPIROPYRAZOLOPYRIDINE DERIVATIVES AND USES THEREOF FOR THE TREATMENT OF VIRAL INFECTIONS NOVARTIS AG (CH) 2014-10-16 WO disclosed