SCHEMBL11483545

SCHEMBL11483545

CC(c1ccc(C(F)(F)F)cc1)n1cnc(C(=O)O)c1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.41
PDE2A O00408 5/20 0.38
ALDH1A1 P00352 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GSK3B P49841 1/20 0.38
TEAD1 P28347 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
PTGER4 P35408 1/20 0.36
IGFBP3 P17936 1/20 0.36
DPP4 P27487 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
BRD4 O60885 1/20 0.36
SRD5A2 P31213 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11491038 0.85 CES2 (0.46) CES2ALDH1A1BRD4
SCHEMBL11483551 0.82 PKM (0.41) PTGDR2ALDH1A1TDP1GAAPKM
SCHEMBL11483998 0.76 PKM (0.39) ALDH1A1TDP1GAAPKMTSHR
SCHEMBL11483657 0.76 KMO (0.41) ALDH1A1AKR1C3AKR1C2GAAPKM
SCHEMBL11488916 0.73 ADRA1D (0.47) ALDH1A1TDP1GAAPKMTSHR
SCHEMBL31002588 0.72 GPBAR1 (0.43) ALDH1A1TDP1
SCHEMBL23212270 0.71 ALDH1A1 (0.52) ALDH1A1TDP1TSHRBRD4
SCHEMBL21298733 0.71 ALDH1A1 (0.52) ALDH1A1TDP1TSHRBRD4
SCHEMBL11484432 0.70 PKM (0.69) ALDH1A1GAAPKMTSHRSRD5A2
SCHEMBL16166195 0.70 PDE2A (0.42) CES2CES1PTGDR2PDE2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4185992-A Imidazole derivatives MAY & BAKER LIMITED (GB) 1980-01-29 US disclosed