SCHEMBL16199856

SCHEMBL16199856

CCCN(CCC)c1ncc(C(N)=O)cn1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 3/20 0.49
NNMT P40261 7/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EPHX2 P34913 1/20 0.38
PARP10 Q53GL7 1/20 0.37
AOC3 Q16853 1/20 0.36
HPGDS O60760 1/20 0.36
TSHR P16473 1/20 0.35
MAPT P10636 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771472 0.75 KDM4E (0.67) NNMTSMN1; SMN2KDM4EALDH1A1ALOX15
SCHEMBL22401242 0.72 NNMT (0.42) HCAR3NNMTSMN1; SMN2KDM4EEPHX2
SCHEMBL5374100 0.71 KDM4E (0.43) HCAR3SMN1; SMN2KDM4EALDH1A1HSD17B10
SCHEMBL12874146 0.71 CRHR1 (0.40) HCAR3SMN1; SMN2ALDH1A1HSD17B10MAPT
SCHEMBL17101820 0.71 NNMT (0.45) NNMTSMN1; SMN2KDM4EEPHX2PARP10
SCHEMBL7257903 0.70 HCAR3 (0.37) HCAR3SMN1; SMN2MAPT
SCHEMBL3121440 0.70 KDM4E (0.46) NNMTSMN1; SMN2KDM4EALDH1A1ALOX15
SCHEMBL14852700 0.70 HCAR3 (0.75) HCAR3NNMTSMN1; SMN2KDM4EEPHX2
SCHEMBL3353364 0.70 HCAR3 (0.48) HCAR3KDM4EHSD17B10PARP10AOC3
SCHEMBL13701705 0.69 KCNA5 (0.44) HCAR3SMN1; SMN2TSHRMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190287-B1 TARTRATE SALTS OR COMPLEXES OF QUINAZOLINE BASED EGFR INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS INC (US) 2014-10-29 EP disclosed