SCHEMBL16200046

SCHEMBL16200046

Cc1ccccc1-c1nn(C)c(C(F)(F)F)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRB2 P47870 1/20 0.39
GABRA4 P48169 1/20 0.39
GABRE P78334 1/20 0.39
GABRA6 Q16445 1/20 0.39
GABRG1 Q8N1C3 1/20 0.39
GABRG3 Q99928 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16200058 0.85 HSD11B1 (0.40) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL14039900 0.80 ALDH1A1 (0.50) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL7524976 0.77 CYP1A2 (0.39) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL14139212 0.76 POLB (0.40) CYP1A2CYP2C19GABRPGABRDGABRA1
SCHEMBL8569766 0.75 HSD11B1 (0.47) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL13682912 0.75 NPC1 (0.41) CYP1A2KDM4EALDH1A1
SCHEMBL8566222 0.73 MEN1 (0.38) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL16200053 0.72 SLC34A1 (0.44) PTGS1PTGS2
SCHEMBL16200057 0.72 MAPK14 (0.42) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL14039556 0.72 NT5E (0.41) CYP1A2PTGS2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed