SCHEMBL16200057

SCHEMBL16200057

Cn1nc(-c2ccncc2)c(Cl)c1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.42
MAPK13 O15264 1/20 0.41
CSNK1D P48730 1/20 0.41
CSNK1E P49674 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
KIF11 P52732 1/20 0.39
ALDH1A1 P00352 2/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 1/20 0.37
BRAF P15056 9/20 0.36
SRC P12931 4/20 0.35
KDR P35968 4/20 0.35
RIPK2 O43353 1/20 0.35
EGFR P00533 1/20 0.35
TNK2 Q07912 1/20 0.35
PTK6 Q13882 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14039900 0.85 ALDH1A1 (0.50) ALDH1A1MAPTHTTKDM4EMEN1
SCHEMBL16200053 0.84 SLC34A1 (0.44) MAPK14MAPK13CSNK1DCSNK1EMAPK12
SCHEMBL16200054 0.82 P2RX7 (0.45) ALDH1A1NPC1RAB9AKDM4ECYP1A2
SCHEMBL16200062 0.80 PTGS2 (0.46) ALDH1A1NPC1MAPTRAB9AKDM4E
SCHEMBL8108697 0.77 SLC34A1 (0.38) ALDH1A1MAPTKDM4EMEN1CYP1A2
SCHEMBL14039556 0.77 NT5E (0.41) ALDH1A1MAPTHTTKDM4ECYP1A2
SCHEMBL16200055 0.76 MAPK14 (0.43) MAPK14MAPK13CSNK1DCSNK1EMAPK12
SCHEMBL13683098 0.74 KIF11 (0.39) MAPK14MAPK13CSNK1DCSNK1EMAPK12
SCHEMBL13682912 0.74 NPC1 (0.41) ALDH1A1NPC1RAB9AKDM4ECYP1A2
SCHEMBL16200046 0.72 MEN1 (0.41) ALDH1A1KDM4EMEN1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed