SCHEMBL16200058

SCHEMBL16200058

Cn1nc(-c2ccccc2F)c(Cl)c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.40
MAPT P10636 5/20 0.39
PDE10A Q9Y233 2/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
MBNL1 Q9NR56 1/20 0.38
TP53 P04637 2/20 0.38
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16200046 0.85 MEN1 (0.41) HSD11B1MEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8569766 0.84 HSD11B1 (0.47) HSD11B1MAPTMEN1CYP1A2CYP2C9
SCHEMBL16200051 0.81 PTGS2 (0.39) HSD11B1MAPTMBNL1TP53ADORA2A
SCHEMBL16200388 0.80 THRB (0.45) HSD11B1MAPTPDE10AKMT2AMBNL1
SCHEMBL14039900 0.80 ALDH1A1 (0.50) MAPTMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8566222 0.79 MEN1 (0.38) HSD11B1MAPTPDE10AMEN1CYP1A2
SCHEMBL27321857 0.78 HSD11B1 (0.43) HSD11B1MAPTMEN1CYP1A2CYP2C9
SCHEMBL13738167 0.77 MAPT (0.40) HSD11B1MAPTMEN1KMT2AMBNL1
SCHEMBL8570221 0.77 MEN1 (0.37) HSD11B1PDE10AMEN1CYP1A2CYP2C9
SCHEMBL8565103 0.77 MEN1 (0.37) HSD11B1MEN1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed