SCHEMBL16212908

SCHEMBL16212908

CN(C(=O)O)n1cnc(-c2ccccc2F)c1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
USP19 O94966 4/20 0.45
GRIN2B Q13224 5/20 0.40
POLB P06746 1/20 0.40
ADORA2A P29274 3/20 0.39
ADORA3 P0DMS8 2/20 0.39
ADORA1 P30542 2/20 0.39
ADORA2B P29275 1/20 0.39
KIF11 P52732 3/20 0.38
NPC1 O15118 1/20 0.38
LTB4R Q15722 1/20 0.38
MAPT P10636 1/20 0.38
DHODH Q02127 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL426697 0.77 FAAH (0.44) USP19GRIN2BPOLBADORA2AADORA3
SCHEMBL427489 0.73 FAAH (0.40) USP19GRIN2BADORA2AADORA3ADORA1
SCHEMBL2731600 0.72 CYP2A6 (0.56)
SCHEMBL15511383 0.70 LMNA (0.33) POLB
SCHEMBL27859118 0.67 MAOA (0.45) POLBNPC1MAPT
SCHEMBL29106080 0.65 ACMSD (0.54) POLBDHODH
SCHEMBL6223694 0.65 KMO (0.54) ADORA2AADORA3ADORA1ADORA2BNPC1
SCHEMBL16566651 0.64 PARP1 (0.39) ADORA2AADORA3ADORA1ADORA2BNPC1
SCHEMBL6028461 0.64 FAAH (0.47) GRIN2BADORA2AADORA3ADORA1ADORA2B
SCHEMBL4498726 0.63 KDM4C (0.64)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991989-A1 IMIDAZO-TRIAZINE DERIVATIVES AS PDE10 INHIBITORS Pfizer Inc. (US) 2016-03-09 EP disclosed
WO-2014177977-A1 IMIDAZO-TRIAZINE DERIVATIVES AS PDE10 INHIBITORS PFIZER INC. (US) 2014-11-06 WO disclosed