SCHEMBL16229756

SCHEMBL16229756

CN1C2C1C21Cc2cc(F)c(CCNS(=O)(=O)CC3CC3)cc2C1Cc1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 4/20 0.32
OPRL1 P41146 1/20 0.32
TBXA2R P21731 2/20 0.31
KCNH2 Q12809 1/20 0.31
RORC P51449 1/20 0.30
EPHX2 P34913 1/20 0.30
ALDH1A1 P00352 1/20 0.30
AKR1C3 P42330 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16229799 0.92 SLC6A9 (0.33) SLC6A9KCNH2
SCHEMBL16229764 0.92 KMT2A (0.32) SLC6A9OPRL1RORC
SCHEMBL16229782 0.91 SLC6A9 (0.39) SLC6A9KCNH2ALDH1A1
SCHEMBL16229802 0.89 GALR3 (0.38) SLC6A9
SCHEMBL16229807 0.88 SLC6A9 (0.36) SLC6A9TBXA2RKCNH2EPHX2ALDH1A1
SCHEMBL16229769 0.88 DPP4 (0.34) SLC6A9RORC
SCHEMBL16229765 0.87 SLC6A9 (0.38) SLC6A9KCNH2
SCHEMBL16229762 0.84 KMT2A (0.32) SLC6A9
SCHEMBL16229761 0.83 SLC6A9 (0.37) SLC6A9TBXA2RALDH1A1AKR1C3
SCHEMBL16784656 0.83 SLC6A9 (0.35) SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051280-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2015-06-09 US disclosed
US-8883839-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy ABBOTT LABORATORIES (US) 2014-11-11 US disclosed