SCHEMBL16229776

SCHEMBL16229776

CN1C2C1C21Cc2ccc(CCNS(=O)(=O)C3CCC3)cc2C1Cc1cccc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.36
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
TP53 P04637 2/20 0.34
MDM2 Q00987 2/20 0.34
TAAR1 Q96RJ0 2/20 0.33
TBXA2R P21731 2/20 0.33
ADRB3 P13945 2/20 0.33
EPHX2 P34913 1/20 0.33
GLA P06280 1/20 0.33
AKR1C3 P42330 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
MAPT P10636 1/20 0.33
SLC2A1 P11166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16784631 0.92 DPP4 (0.36) SLC6A9DPP4DPP8DPP9DPP7
SCHEMBL16229755 0.91 TBXAS1 (0.36) SLC6A9TAAR1
SCHEMBL16229775 0.90 DGAT1 (0.36) SLC6A9TAAR1MAPT
SCHEMBL16229771 0.88 GALR3 (0.38) SLC6A9DPP4
SCHEMBL16229807 0.87 SLC6A9 (0.36) SLC6A9TAAR1TBXA2REPHX2GLA
SCHEMBL16784646 0.87 SLC6A9 (0.49) SLC6A9
SCHEMBL16229769 0.87 DPP4 (0.34) SLC6A9DPP4DPP8DPP9DPP7
SCHEMBL16229805 0.83 SLC6A9 (0.38) SLC6A9DPP4DPP8DPP9DPP7
SCHEMBL16229783 0.82 SLC6A9 (0.41) SLC6A9TBXA2RAKR1C3MAPT
SCHEMBL16784656 0.82 SLC6A9 (0.35) SLC6A9TP53CNR1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051280-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2015-06-09 US disclosed
US-8883839-B2 Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy ABBOTT LABORATORIES (US) 2014-11-11 US disclosed