SCHEMBL16234635

SCHEMBL16234635

COc1ccc2ccn(CC(C)=O)c2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.65
MTNR1B P49286 6/20 0.65
HTR2A P28223 1/20 0.57
HTR2C P28335 1/20 0.57
MCL1 Q07820 1/20 0.52
HDAC8 Q9BY41 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
TRPV1 Q8NER1 1/20 0.50
HTR7 P34969 1/20 0.49
MAOA P21397 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10222047 0.88 MTNR1A (0.61) MTNR1AMTNR1BHTR2AHTR2CMCL1
SCHEMBL6099343 0.87 MTNR1A (0.60) MTNR1AMTNR1BHTR2AHTR2CMCL1
SCHEMBL11984620 0.85 MTNR1A (0.63) MTNR1AMTNR1BHTR2AHTR2CMCL1
SCHEMBL10165374 0.84 MTNR1A (0.57) MTNR1AMTNR1BHTR2AHTR2CMCL1
SCHEMBL10204441 0.81 MTNR1A (0.55) MTNR1AMTNR1BHTR2AHTR2CMCL1
SCHEMBL980885 0.79 HTR2C (0.65) MTNR1AMTNR1BHTR2AHTR2CMCL1
SCHEMBL16543633 0.78 ALDH1A1 (0.48) MTNR1AMTNR1BKDM4ESMN1; SMN2LMNA
SCHEMBL13139567 0.78 NTSR1 (0.45) MTNR1AMTNR1BHTR2AHTR2CKDM4E
SCHEMBL12605655 0.78 FKBP1A (0.53) MTNR1AMTNR1BHTR2AHTR2CHTR7
SCHEMBL9701534 0.77 KMT2A (0.71) HTR2AHTR2CHDAC8HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8883766-B2 Ion channel modulators and methods of use VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-11-11 US disclosed