SCHEMBL16239479

SCHEMBL16239479

CC1(C)CC(c2cccc(NS(=O)(=O)c3ccccc3F)c2)Nc2c(C#N)cccc21

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
KDM1A O60341 4/20 0.38
KMT2A Q03164 1/20 0.38
SLC22A12 Q96S37 9/20 0.37
BRD1 O95696 1/20 0.37
BRPF1 P55201 1/20 0.37
CASP3 P42574 1/20 0.37
NLRP3 Q96P20 1/20 0.36
MAOB P27338 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239989 0.87 IMPDH2 (0.40) BRD4KDM1AKMT2A
SCHEMBL16239497 0.87 L3MBTL1 (0.43) BRD4KMT2A
SCHEMBL16239598 0.87 KMT2A (0.39) KMT2A
SCHEMBL16239646 0.86 BRD4 (0.40) BRD4KMT2ACASP3NLRP3
SCHEMBL16239481 0.86 BRD4 (0.36) BRD4KDM1A
SCHEMBL16240123 0.85 SLC22A12 (0.43) BRD4SLC22A12CASP3NLRP3
SCHEMBL16240087 0.84 GPR119 (0.41) BRD4KMT2A
SCHEMBL2135474 0.83 BRD4 (0.42) BRD4KMT2ASLC22A12CASP3NLRP3
SCHEMBL2134891 0.79 BRD4 (0.44) BRD4KMT2ACASP3NLRP3
SCHEMBL2136761 0.79 BRD4 (0.43) BRD4KMT2ACASP3NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630124-B1 TETRAHYDROQUINOLINE DERIVATIVES USED AS AMPK ACTIVATORS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed