SCHEMBL16239481

SCHEMBL16239481

CC1(C)CC(c2cccc(NS(C)(=O)=O)c2)Nc2c(C#N)cccc21

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.36
CREBBP Q92793 1/20 0.36
CSNK2A2 P19784 1/20 0.36
OPRM1 P35372 1/20 0.35
KDM1A O60341 1/20 0.35
F11 P03951 1/20 0.35
F7 P08709 1/20 0.35
ALDH1A1 P00352 2/20 0.33
TDP2 O95551 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
PGR P06401 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSP90AA1 P07900 3/20 0.33
HSP90AB1 P08238 3/20 0.33
HRH3 Q9Y5N1 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239989 0.89 IMPDH2 (0.40) BRD4KDM1AALDH1A1LMNASMN1; SMN2
SCHEMBL16240087 0.88 GPR119 (0.41) BRD4ALDH1A1LMNASMN1; SMN2
SCHEMBL16239598 0.87 KMT2A (0.39) ALDH1A1LMNAPGRPOLB
SCHEMBL16239497 0.87 L3MBTL1 (0.43) BRD4ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL16239479 0.86 BRD4 (0.38) BRD4KDM1A
SCHEMBL16239494 0.85 BRD4 (0.39) BRD4CREBBPOPRM1KDM1AF11
SCHEMBL16239477 0.84 BRD4 (0.38) BRD4CREBBPOPRM1KDM1AF11
SCHEMBL16239647 0.81 PLA2G7 (0.37) CSNK2A2
SCHEMBL16239667 0.81 KIF11 (0.40) BRD4CREBBPOPRM1KDM1AF11
SCHEMBL2134882 0.80 F11 (0.41) BRD4CREBBPCSNK2A2OPRM1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630124-B1 TETRAHYDROQUINOLINE DERIVATIVES USED AS AMPK ACTIVATORS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed