SCHEMBL16239598

SCHEMBL16239598

CC1(C)CC(c2cccc(NS(=O)(=O)c3cccc(F)c3)c2)Nc2c(C#N)cccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
HTR1A P08908 2/20 0.37
HTR2C P28335 2/20 0.37
HTR7 P34969 2/20 0.37
HTR6 P50406 2/20 0.37
MOGAT2 Q3SYC2 1/20 0.37
HSD11B1 P28845 1/20 0.37
ALDH1A1 P00352 1/20 0.36
ESR1 P03372 1/20 0.36
MAPT P10636 4/20 0.36
TP53 P04637 3/20 0.36
LMNA P02545 2/20 0.36
PGR P06401 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
AURKA O14965 1/20 0.35
KDR P35968 1/20 0.35
AURKB Q96GD4 1/20 0.35
SLC10A2 Q12908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16239497 0.93 L3MBTL1 (0.43) KMT2AMOGAT2HSD11B1ALDH1A1ESR1
SCHEMBL16239989 0.92 IMPDH2 (0.40) KMT2AHTR6ALDH1A1MAPTLMNA
SCHEMBL16240087 0.88 GPR119 (0.41) KMT2AALDH1A1ESR1MAPTTP53
SCHEMBL16239481 0.87 BRD4 (0.36) POLBALDH1A1LMNAPGR
SCHEMBL16239479 0.87 BRD4 (0.38) KMT2A
SCHEMBL16239627 0.86 KMT2A (0.41) KMT2APOLBPKMHSD11B1ALDH1A1
SCHEMBL2133368 0.83 PKM (0.41) KMT2APOLBPKMHTR6HSD11B1
SCHEMBL2136004 0.79 PKM (0.44) KMT2APOLBPKMHSD11B1ALDH1A1
SCHEMBL16240075 0.79 L3MBTL1 (0.45) KMT2AHSD11B1ALDH1A1ESR1MAPT
SCHEMBL16239486 0.78 HPGD (0.43) KMT2AHTR6ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630124-B1 TETRAHYDROQUINOLINE DERIVATIVES USED AS AMPK ACTIVATORS HOFFMANN LA ROCHE (CH) 2014-11-19 EP claimed