SCHEMBL16247338

SCHEMBL16247338

CC1(C)OB(c2ccc(COC(=O)NCc3ccccc3C(=O)O)cc2)OC1(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
KCNA5 P22460 8/20 0.45
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
PLAU P00749 1/20 0.40
KCNK3 O14649 1/20 0.40
KCNA3 P22001 1/20 0.40
LPL P06858 1/20 0.39
LIPG Q9Y5X9 1/20 0.39
DGAT1 O75907 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9986887 0.91 KEAP1 (0.43) KEAP1NFE2L2KCNA5CA1CA2
SCHEMBL14934909 0.87 KEAP1 (0.55) KEAP1NFE2L2CA1CA2CA9
SCHEMBL16030765 0.87 KEAP1 (0.55) KEAP1NFE2L2CA1CA2CA9
SCHEMBL6989373 0.81 KCNA5 (0.57) KEAP1NFE2L2KCNA5PLAUKCNK3
SCHEMBL28659356 0.81 CA1 (0.55) KEAP1NFE2L2KCNA5CA1CA2
SCHEMBL25217470 0.81 L3MBTL1 (0.42) KEAP1NFE2L2KCNA5PLAULIPG
SCHEMBL29707329 0.80 CA2 (0.52) KEAP1NFE2L2CA1CA2CA9
SCHEMBL29707332 0.80 CA2 (0.52) KEAP1NFE2L2CA1CA2CA9
SCHEMBL24142282 0.79 LIPG (0.54) KEAP1NFE2L2CA1CA2CA9
SCHEMBL30543686 0.77 HTT (0.51) KEAP1NFE2L2CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889638-B2 Stimulus-triggered prodrugs THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-11-18 US disclosed