SCHEMBL16257540

SCHEMBL16257540

COc1cc(/C=C/C(=O)c2cccc(N)c2)cc(OC)c1O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.65
ABCG2 Q9UNQ0 4/20 0.63
NPC1 O15118 1/20 0.63
PTPN1 P18031 1/20 0.62
NR1H4 Q96RI1 1/20 0.60
CA1 P00915 2/20 0.59
CA2 P00918 2/20 0.59
KRAS P01116 1/20 0.59
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2B6 P20813 1/20 0.56
LMNA P02545 2/20 0.56
MAPT P10636 2/20 0.56
HTT P42858 2/20 0.56
GAA P10253 1/20 0.56
PKM P14618 1/20 0.55
PTGS1 P23219 1/20 0.55
PTGS2 P35354 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14760794 0.90 ABCB1 (0.82) ABCB1ABCG2CA1CA2KRAS
SCHEMBL14760795 0.90 ABCB1 (0.82) ABCB1ABCG2CA1CA2KRAS
SCHEMBL2221923 0.87 RELA (0.68) PTPN1NR1H4CA1CA2PTGS1
SCHEMBL2221920 0.87 RELA (0.68) PTPN1NR1H4CA1CA2PTGS1
SCHEMBL16257539 0.87 NR1H4 (0.74) ABCB1ABCG2NR1H4CA1CA2
SCHEMBL29803052 0.87 NR1H4 (0.74) ABCB1ABCG2NR1H4CA1CA2
SCHEMBL7096493 0.82 ABCG2 (0.70) ABCB1ABCG2NPC1PTPN1NR1H4
SCHEMBL16597316 0.81 ABCG2 (0.72) ABCG2NPC1CYP1A2CYP3A4CYP2D6
SCHEMBL16597306 0.81 ABCG2 (0.72) ABCG2NPC1CYP1A2CYP3A4CYP2D6
SCHEMBL7096880 0.80 NR1H4 (0.74) ABCB1NPC1PTPN1NR1H4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8889874-B2 Imidazolone-chalcone derivatives as potential anticancer agent and process for the preparation thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2014-11-18 US disclosed