SCHEMBL16265367

SCHEMBL16265367

COc1ccccc1NC(=O)Nc1ccccc1NS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
TSHR P16473 1/20 0.65
HTT P42858 2/20 0.62
MEN1 O00255 4/20 0.60
KMT2A Q03164 4/20 0.60
ALDH1A1 P00352 2/20 0.60
POLB P06746 1/20 0.60
CA12 O43570 2/20 0.58
CA1 P00915 2/20 0.58
CA2 P00918 2/20 0.58
CA9 Q16790 2/20 0.58
MAPT P10636 5/20 0.57
MAPK1 P28482 1/20 0.57
KDM4E B2RXH2 2/20 0.55
GAA P10253 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572319 0.86 POLB (0.68) LMNASMN1; SMN2HTTMEN1KMT2A
SCHEMBL23200304 0.85 KMT2A (0.67) LMNASMN1; SMN2TSHRHTTMEN1
SCHEMBL17102981 0.84 SMN1; SMN2 (0.61) LMNASMN1; SMN2TSHRHTTMEN1
SCHEMBL16672112 0.84 LMNA (0.72) LMNASMN1; SMN2TSHRHTTMEN1
SCHEMBL16290773 0.83 MAPT (0.60) LMNASMN1; SMN2TSHRHTTMEN1
SCHEMBL15145840 0.83 LMNA (0.70) LMNASMN1; SMN2TSHRHTTMEN1
SCHEMBL20568014 0.82 ALDH1A1 (0.65) LMNASMN1; SMN2TSHRHTTMEN1
SCHEMBL20567802 0.82 LMNA (0.74) LMNASMN1; SMN2TSHRKMT2AALDH1A1
SCHEMBL30343051 0.82 MAPT (0.58) LMNASMN1; SMN2HTTMEN1KMT2A
SCHEMBL23141078 0.82 MAPT (0.58) LMNASMN1; SMN2HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9216954-B2 Serine racemase inhibitor NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2015-12-22 US disclosed
US-9216954-B2 Serine racemase inhibitor NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2015-12-22 US disclosed
US-20140371291-A1 SERINE RACEMASE INHIBITOR NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2014-12-18 US disclosed
US-20140371291-A1 SERINE RACEMASE INHIBITOR NATIONAL UNIVERSITY CORPORATION UNIVERSITY OF TOYAMA (JP) 2014-12-18 US disclosed
EP-2808014-A1 SERINE RACEMASE INHIBITOR National University Corporation University Of Toyama (JP) 2014-12-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140371291-A1 SERINE RACEMASE INHIBITOR SRR, PRSS1, ME1 LMNA 3748/4885SMN1; SMN2 967/4885TSHR 4233/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.