SCHEMBL16269151

SCHEMBL16269151

O=C(O)COc1cccc2c1CN(C(=O)O)CC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.53
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
NOTUM Q6P988 1/20 0.47
POLB P06746 1/20 0.45
PARP1 P09874 1/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 2/20 0.45
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
CD69 Q07108 1/20 0.44
S1PR5 Q9H228 4/20 0.43
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28864977 0.89 ABHD6 (0.49) PTGDR2ALDH1A1MEN1KMT2ANOTUM
SCHEMBL16268884 0.84 PTGDR2 (0.52) PTGDR2ALDH1A1MEN1KMT2ANOTUM
SCHEMBL28534873 0.83 HRH3 (0.47) PTGDR2MEN1KMT2ANOTUMHPGD
SCHEMBL30641865 0.82 DRD2 (0.51) KMT2ANOTUMHSD17B10KDM4E
SCHEMBL19599364 0.81 ADRA2A (0.60) ALDH1A1S1PR5PRMT5WDR77RXRA
SCHEMBL3479749 0.77 RXRB (0.66) POLBHSD17B10KDM4ECD69TSHR
SCHEMBL28245905 0.76 TAAR1 (0.40) ALDH1A1MEN1KMT2ANOTUMPARP1
SCHEMBL28548896 0.76 RXRB (0.64) PTGDR2POLBHSD17B10KDM4ECD69
SCHEMBL18586143 0.75 PTGDR2 (0.41) PTGDR2ALDH1A1KMT2AHPGDHSD17B10
SCHEMBL30726807 0.75 ALDH1A1 (0.51) PTGDR2ALDH1A1MEN1KMT2ANOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105263924-B Cxcr7 receptor modulators 爱杜西亚制药有限公司 2018-10-19 CN disclosed
EP-3004082-A1 CXCR7 RECEPTOR MODULATORS Actelion Pharmaceuticals Ltd. (CH) 2016-04-13 EP disclosed
WO-2014191929-A1 CXCR7 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2014-12-04 WO disclosed