SCHEMBL1628

SCHEMBL1628

COC(=O)C(C)CN(C)c1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.43
MME P08473 1/20 0.42
FFAR1 O14842 1/20 0.42
AKR1B1 P15121 1/20 0.42
PTPN5 P54829 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA4 P48058 1/20 0.38
PTPN1 P18031 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
OXTR P30559 3/20 0.37
AVPR1A P37288 3/20 0.37
ITGB1 P05556 1/20 0.37
ITGA4 P13612 1/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MYC P01106 1/20 0.37
WDR5 P61964 1/20 0.37
AVPR2 P30518 1/20 0.36
GAA P10253 2/20 0.36
ALDH1A1 P00352 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270546 0.87 ESR2 (0.46) ESR2MMEFFAR1AKR1B1PTPN5
SCHEMBL2686 0.81 ESR2 (0.40) ESR2MMEFFAR1AKR1B1PTPN5
SCHEMBL7279558 0.79 ESR2 (0.46) ESR2MMEFFAR1AKR1B1PTPN5
SCHEMBL3008 0.78 LTB4R2 (0.50) MMEFFAR1AKR1B1OXTRAVPR1A
SCHEMBL1629 0.77 MYC (0.45) ESR2MMEFFAR1AKR1B1PTPN5
SCHEMBL2104 0.77 NLRP3 (0.43) ESR2MMEFFAR1AKR1B1PTPN5
SCHEMBL14496801 0.74 TDP1 (0.42) MAPK1SMN1; SMN2GAAALDH1A1HPGD
SCHEMBL2870 0.74 MYC (0.47) ESR2MMEFFAR1AKR1B1PTPN5
SCHEMBL2132 0.74 MYC (0.47) ESR2MMEFFAR1AKR1B1PTPN5
SCHEMBL14998792 0.74 AGTR1 (0.44) ESR2MMEFFAR1AKR1B1PTPN5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed