SCHEMBL163055

SCHEMBL163055

CCOC(=O)C(C)N(C(=O)c1ccccc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.45
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
PLA2G1B P04054 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 3/20 0.40
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
POLB P06746 1/20 0.39
PPARG P37231 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8827400 1.00 RORC (0.45) RORCMEN1KMT2AHTTNPSR1
SCHEMBL6294014 1.00 RORC (0.45) RORCMEN1KMT2AHTTNPSR1
SCHEMBL8540022 0.96 RORC (0.43) RORCMEN1KMT2AHTTNPSR1
SCHEMBL11284170 0.89 MEN1 (0.46) RORCMEN1KMT2AHTTNPSR1
Clopyralid SCHEMBL6933656 0.89 L3MBTL1 (0.41) RORCMEN1KMT2AHTTNPSR1
SCHEMBL635894 0.89 RORC (0.43) RORCMEN1KMT2AHTTNPSR1
SCHEMBL635895 0.89 RORC (0.43) RORCMEN1KMT2AHTTNPSR1
SCHEMBL9617379 0.87 KMT2A (0.54) MEN1KMT2AHTTNPSR1PLA2G1B
SCHEMBL10858376 0.85 MEN1 (0.42) RORCMEN1KMT2AHTTNPSR1
SCHEMBL4894608 0.84 CHRM2 (0.45) MEN1KMT2AHTTNPSR1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2122 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
US-20230000079-A1 COMBINATION COMPRISING A TRIKETONE HERBICIDE AND A DIPHENYLETHER HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2023-01-05 US claimed
US-20220015371-A1 Compositions and Methods for Reducing Pesticide-Induced Plant Damage and Improving Plant Yield PNC BANK, NATIONAL ASSOCIATION 2022-01-20 US claimed
US-20210378241-A1 COMBINATION COMPRISING A BENZAMIDE HERBICIDE AND A PYRIDINE CARBOXYLIC ACID HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2021-12-09 US claimed
EP-3890491-A1 COMPOSITIONS AND METHODS FOR REDUCING PESTICIDE-INDUCED PLANT DAMAGE AND IMPROVING PLANT YIELD Cytozyme Laboratories, Inc. (US) 2021-10-13 EP claimed
US-20210120811-A1 AQUEOUS CAPSULE SUSPENSION CONCENTRATES CONTAINING A HERBICIDAL SAFENER AND A PESTICIDAL ACTIVE SUBSTANCE FMC CORPORATION 2021-04-29 US claimed
EP-3787407-A1 AQUEOUS CAPSULE SUSPENSION CONCENTRATES CONTAINING A HERBICIDAL SAFENER AND A PESTICIDAL ACTIVE SUBSTANCE Bayer Aktiengesellschaft (DE) 2021-03-10 EP claimed
US-10897896-B2 High load aqueous suspension concentrate of an active ingredient DOW AGROSCIENCES LLC (US) 2021-01-26 US claimed
EP-3174865-B1 MOLECULES HAVING CERTAIN PESTICIDAL UTILITIES, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES RELATED THERETO DOW AGROSCIENCES LLC (US) 2020-12-09 EP claimed
US-20200236925-A1 METHODS AND FORMULATIONS FOR PREVENTING DOWNWARD MIGRATION OF AGRICULTURAL MATERIALS DISCOVERY PURCHASER CORPORATION 2020-07-30 US claimed
EP-0784431-A1 SYNERGISTIC ACTIVE SUBSTANCE HERBICIDE COMBINATIONS WITH 1-(2,6-DICHLORO-4-DIFLUOROMETHYL-PHENYL)-5-(2-CHLOROPROPIONAMIDO)-4-NITROPYRAZOL BAYER AG (DE) 1997-07-23 EP claimed
WO-1997010714-A1 HERBICIDAL MIXTURES HAVING A SYNERGISTIC EFFECT BASF AKTIENGESELLSCHAFT (DE) 1997-03-27 WO claimed
WO-1996010333-A1 SYNERGISTIC ACTIVE SUBSTANCE HERBICIDE COMBINATIONS WITH 1-(2,6-DICHLORO-4-DIFLUOROMETHYL-PHENYL)-5-(2-CHLOROPROPIONAMIDO)-4-NITROPYRAZOL BAYER AKTIENGESELLSCHAFT (DE) 1996-04-11 WO claimed
US-5223016-A HERBICIDAL COMPOSITIONS COMPRISING BENZOFURYLOXYPHENYLUREA OR BENZOPYRANYLOXYPHENYLUREA HERBICIDES AND DICAMBA, TRICLOPYR, MECOPROP, FLUROXYPYR, BENTAZONE, OR METRIBUZIN MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1993-06-29 US claimed
EP-0448723-A1 HERBICIDAL COMPOSITION AND METHOD OF KILLING WEED MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1991-10-02 EP claimed
EP-0434613-A2 Synergistic agent and method of regulating plant growth CIBA-GEIGY AG (CH) 1991-06-26 EP claimed
EP-0113857-A1 Herbicidal agents BAYER AG (DE) 1984-07-25 EP claimed
EP-0052825-A1 Selective herbicidal agents on the basis of triazine diones BAYER AG (DE) 1982-06-02 EP claimed
EP-0005917-A1 Herbicidal method and mixtures of herbicidal heterocyclic compounds FISONS plc (GB) 1979-12-12 EP claimed
US-3976468-A Herbicide mixture of lower alkyl esters of N-benzoyl-N-chlorophenyl-2-amino-lower alkanoic acids and 3-lower alkyl-2,1,3-benzothiadiazinone-(4)-2,2-dioxides or salts thereof BASF AKTIENGESELLSCHAFT (DT) 1976-08-24 US claimed