SCHEMBL1632043

SCHEMBL1632043

Cc1cccc(CCNc2nc(-c3ccccc3)ccc2C(C(N)=O)c2cccnc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
CYP1A2 P05177 3/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C19 P33261 3/20 0.40
MAPT P10636 3/20 0.40
KDM4E B2RXH2 3/20 0.40
HSD17B10 Q99714 2/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
HIF1A Q16665 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PTAFR P25105 1/20 0.40
JAK3 P52333 1/20 0.39
GBA1 P04062 4/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1631443 0.91 NPC1 (0.45) ALDH1A1MAPTMEN1KMT2AGBA1
SCHEMBL1631415 0.90 GBA1 (0.45) ALDH1A1MAPTMEN1KMT2APTAFR
SCHEMBL1630102 0.90 CSNK2A2 (0.44) ALDH1A1MAPTMEN1KMT2AHIF1A
SCHEMBL1631787 0.90 GBA1 (0.51) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL1632284 0.89 CSNK2A2 (0.46) CYP1A2CYP3A4CYP2D6CYP2C19MAPT
SCHEMBL1630481 0.88 CYP3A4 (0.41) ALDH1A1CYP1A2CYP3A4CYP2C19MAPT
SCHEMBL4120643 0.88 ALDH1A1 (0.42) ALDH1A1MAPTKDM4EMEN1LMNA
SCHEMBL1629879 0.86 GBA1 (0.39) ALDH1A1MAPTGBA1SMN1; SMN2NPC1
SCHEMBL1631828 0.86 GBA1 (0.42) ALDH1A1MAPTKDM4ELMNATSHR
SCHEMBL1632985 0.86 ADRB3 (0.42) ALDH1A1MAPTGBA1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090012126-A1 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. 2009-01-08 US claimed
US-7932270-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2011-04-26 US disclosed
US-20090012126-A1 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. 2009-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012126-A1 Certain chemical entities, compositions, and methods MYLK, MYH2, MYH10 ALDH1A1 1756/4885CYP1A2 1688/4885CYP3A4 2030/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.