SCHEMBL1632066

SCHEMBL1632066

N#Cc1ccccc1-c1ccc(N(C=O)Cc2cc[nH]n2)c(NCCc2cccc(F)c2)n1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.34
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KDM4E B2RXH2 1/20 0.31
GBA1 P04062 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
ADORA2A P29274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1629932 0.88 KDM4E (0.43) GPR84NPC1RAB9AKDM4EGBA1
SCHEMBL1630790 0.87 GBA1 (0.35) GPR84NPC1RAB9AKDM4EGBA1
SCHEMBL1632788 0.87 GRM5 (0.36) GPR84NPC1RAB9AKDM4EGBA1
SCHEMBL1630876 0.87 KDM4E (0.33) GPR84NPC1RAB9AKDM4EGBA1
SCHEMBL1632416 0.86 GPR84 (0.37) GPR84KDM4EGBA1LMNAMAPT
SCHEMBL1631283 0.86 GBA1 (0.37) NPC1RAB9AKDM4EGBA1LMNA
SCHEMBL1630804 0.86 CCNC (0.34) GPR84NPC1RAB9AKDM4EGBA1
SCHEMBL1630961 0.86 GABRA1 (0.33) GPR84KDM4EGBA1LMNAMAPT
SCHEMBL1631033 0.85 ADORA2A (0.35) GPR84NPC1RAB9AKDM4EGBA1
SCHEMBL1631221 0.85 ADORA2A (0.34) GPR84NPC1RAB9AKDM4EGBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090012126-A1 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. 2009-01-08 US claimed
US-7932270-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2011-04-26 US disclosed
US-20090012126-A1 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. 2009-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012126-A1 Certain chemical entities, compositions, and methods MYLK, MYH2, MYH10 GPR84 1432/4885NPC1 4711/4885RAB9A 1811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.