SCHEMBL1633737

SCHEMBL1633737

CC(C)(C)[C@@]1(C)CN(Cc2cccc(-c3cccc(CN)c3)n2)CCN1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 2/20 0.39
KLK1 P06870 2/20 0.39
CHRM3 P20309 1/20 0.36
CFD P00746 3/20 0.36
ACACB O00763 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
ACACA Q13085 1/20 0.34
KARS1 Q15046 1/20 0.33
WNK1 Q9H4A3 1/20 0.33
MTOR P42345 1/20 0.33
PLAU P00749 2/20 0.32
PLG P00747 1/20 0.32
PLAT P00750 1/20 0.32
ABL1 P00519 1/20 0.32
USP19 O94966 1/20 0.32
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1362390 0.86 FAAH (0.41) KLKB1KLK1CHRM3CFDPARP1
SCHEMBL1362605 0.85 LOXL2 (0.40) CFDWNK1USP19CNR2
SCHEMBL1632745 0.81 KLK1 (0.40) KLKB1KLK1CHRM3CFDCYP3A4
SCHEMBL1365235 0.79 CHRM3 (0.40) CHRM3
SCHEMBL3411496 0.79 CHRM3 (0.40) CHRM3
SCHEMBL1632056 0.78 FAAH (0.48) CHRM3
SCHEMBL1631726 0.77 CYP2E1 (0.40) KLKB1KLK1CHRM3CYP3A4CYP2C9
SCHEMBL1632732 0.76 SLC2A1 (0.38) CHRM3
SCHEMBL4052726 0.76 CHRM3 (0.45) KLKB1KLK1CHRM3CFDKARS1
SCHEMBL1363928 0.74 CHRM3 (0.39) CHRM3WNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7932247-B2 M3 muscarinic acetylcholine receptor antagonists GLAXO GROUP LIMITED (GB) 2011-04-26 US disclosed