SCHEMBL16352144

SCHEMBL16352144

CC(=O)N(CCC[PH](=O)O)OCc1ccc2ccccc2c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.38
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 1/20 0.37
CYP1A2 P05177 1/20 0.37
MAOB P27338 1/20 0.37
MC4R P32245 1/20 0.36
MC3R P41968 1/20 0.36
KCNH2 Q12809 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
TACR1 P25103 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16352111 0.85 L3MBTL1 (0.45) MAOB
SCHEMBL16352145 0.83 L3MBTL1 (0.40) RAB9A
SCHEMBL16352150 0.83 ATM (0.44) MAOBRAB9AATM
SCHEMBL16352147 0.82 NR4A2 (0.40)
SCHEMBL16352154 0.81 MAOB (0.38) CYP1A2MAOBRAB9AATM
SCHEMBL16352153 0.81 MAOB (0.43) MAOB
SCHEMBL16363847 0.81 MME (0.42) SIGMAR1SLC1A3SLC1A2SLC1A1SLC6A2
SCHEMBL16352121 0.81 SLC1A3 (0.40) SIGMAR1SLC1A3SLC1A2SLC1A1SLC6A2
SCHEMBL10617048 0.81 SIGMAR1 (0.52) SIGMAR1CYP1A2MC4RMC3RHDAC1
SCHEMBL16352143 0.81 RXRA (0.39) RAB9AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9593136-B2 Compounds for inhibiting 1-deoxy-D-xylulose-5-phosphate reductoisomerase THE GEORGE WASHINGTON UNIVERSITY (US) 2017-03-14 US disclosed
US-20140378418-A1 COMPOUNDS FOR INHIBITING 1-DEOXY-D-XYLULOSE-5-PHOSPHATE REDUCTOISOMERASE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 2014-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140378418-A1 COMPOUNDS FOR INHIBITING 1-DEOXY-D-XYLULOSE-5-PHOSPHATE REDUCTOISOMERASE DCXR, G6PD, GRHPR SIGMAR1 935/4885SLC1A3 3736/4885SLC1A2 3487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.