SCHEMBL163825

SCHEMBL163825

O=C(O)C1CC(O)C(O)C(O)C1O

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRR1 P24046 3/20 0.43
SLC1A2 P43004 3/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GRM8 O00222 1/20 0.39
GRM6 O15303 1/20 0.39
LMNA P02545 1/20 0.39
APEX1 P27695 1/20 0.39
GRM5 P41594 1/20 0.39
PMP22 Q01453 1/20 0.39
GRM1 Q13255 1/20 0.39
GRM2 Q14416 1/20 0.39
GRM3 Q14832 1/20 0.39
GRM4 Q14833 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC1A1 P43005 2/20 0.38
GABRR2 P28476 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18253254 1.00 GABRR1 (0.43) GABRR1SLC1A2CYP2C9CYP2C19GRM8
SCHEMBL16380722 1.00 GABRR1 (0.43) GABRR1SLC1A2CYP2C9CYP2C19GRM8
SCHEMBL17484815 1.00 GABRR1 (0.43) GABRR1SLC1A2CYP2C9CYP2C19GRM8
SCHEMBL30756696 1.00 GABRR1 (0.43) GABRR1SLC1A2CYP2C9CYP2C19GRM8
SCHEMBL28265022 0.88
SCHEMBL14191347 0.81 GABRR1 (0.42) GABRR1SLC1A2SLC1A1GABRR2
SCHEMBL22602662 0.81 GABRR1 (0.42) GABRR1SLC1A2SLC1A1GABRR2
SCHEMBL19762835 0.81 GABRR1 (0.42) GABRR1SLC1A2SLC1A1GABRR2
SCHEMBL4083282 0.79 GABRR1 (0.50) GABRR1SLC1A2CYP2C9CYP2C19GRM8
SCHEMBL3742301 0.79 GABRR1 (0.50) GABRR1SLC1A2CYP2C9CYP2C19GRM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10342777-B2 Caffeoylquinic acid-rich extract and preparation as well as use thereof MACAU UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2019-07-09 US disclosed
US-20180002275-A1 HYPDH INHIBITORS AND METHODS OF USE FOR THE TREATMENT OF KIDNEY STONES WAKE FOREST UNIVERSITY HEALTH SCIENCES 2018-01-04 US disclosed
US-20170095443-A1 CAFFEOYLQUINIC ACID-RICH EXTRACT AND PREPARATION AS WELL AS USE THEREOF MACAU UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2017-04-06 US disclosed
US-20150038668-A1 Branched Polyesters Based On Citric Acid, Their Preparation And Use BASF SE (DE) 2015-02-05 US disclosed
EP-2611852-B1 BRANCHED POLYESTERS BASED ON CITRIC ACID AND ALSO THEIR PREPARATION AND USE BASF SE (DE) 2014-07-30 EP disclosed
EP-2611852-A1 BRANCHED POLYESTERS BASED ON CITRIC ACID AND ALSO THEIR PREPARATION AND USE BASF SE (DE) 2013-07-10 EP disclosed
WO-2012028496-A1 BRANCHED POLYESTERS BASED ON CITRIC ACID AND ALSO THEIR PREPARATION AND USE BASF SE (DE) 2012-03-08 WO disclosed
EP-2118079-A1 SYNTHETIC MACROCYCLIC COMPOUNDS FOR TREATING CANCER The Government of the United States of America as represented by the Secretary of the Department of Health and Human Services (US) 2009-11-18 EP disclosed
WO-2008098138-A1 SYNTHETIC MACROCYCLIC COMPOUNDS FOR TREATING CANCER THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2008-08-14 WO disclosed
CN-101142211-A Process and method for preparing optically active cis-2-hydroxymethyl-4- (cytosin-1' -yl) -1, 3-oxathiolane or pharmaceutically acceptable salts thereof SERRE BIOLOG CHEMISTRY COMPANY (CA) 2008-03-12 CN disclosed
EP-1009398-A4 MOLECULAR COMPLEX AND CONTROL-RELEASE OF ALPHA HYDROXYACIDS YU RUEY J (US) 2004-06-23 EP disclosed
EP-1009398-A1 MOLECULAR COMPLEX AND CONTROL-RELEASE OF ALPHA HYDROXYACIDS Yu, Ruey J., Dr. (US) 2000-06-21 EP disclosed
WO-1998046217-A1 MOLECULAR COMPLEX AND CONTROL-RELEASE OF ALPHA HYDROXYACIDS YU RUEY J (US) 1998-10-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170095443-A1 CAFFEOYLQUINIC ACID-RICH EXTRACT AND PREPARATION AS WELL AS USE THEREOF CHCHD6, FABP3, TNNT2 GABRR1 540/4885SLC1A2 1196/4885CYP2C9 1687/4885
US-20180002275-A1 HYPDH INHIBITORS AND METHODS OF USE FOR THE TREATMENT OF KIDNEY STONES XDH, GLS, GRHPR GABRR1 1840/4885SLC1A2 1748/4885CYP2C9 633/4885
US-10342777-B2 Caffeoylquinic acid-rich extract and preparation as well as use thereof CHCHD6, FABP3, TNNT2 GABRR1 540/4885SLC1A2 1196/4885CYP2C9 1687/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.