SCHEMBL16396342

SCHEMBL16396342

Nc1ccc2sc(C(=O)O)c(O)c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 3/20 0.45
MAPT P10636 4/20 0.42
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP3A4 P08684 2/20 0.42
MEN1 O00255 2/20 0.42
THRB P10828 2/20 0.42
RECQL P46063 2/20 0.42
KMT2A Q03164 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
HPGD P15428 2/20 0.42
TNF P01375 1/20 0.42
HSPD1 P10809 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
CYP2C19 P33261 1/20 0.42
PTGS2 P35354 1/20 0.42
KDR P35968 1/20 0.42
BRCA1 P38398 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1066852 0.81 GPR35 (0.58) GPR35MAPTALDH1A1KDM4ECYP3A4
SCHEMBL16395952 0.81 KDM4E (0.54) MAPTALDH1A1KDM4EMEN1KMT2A
SCHEMBL17173228 0.79 MCL1 (0.55) GPR35MAPTMEN1KMT2AMCL1
SCHEMBL15697527 0.76 G6PD (0.43) GPR35ALDH1A1KDM4EHPGDCYP2C9
SCHEMBL11804710 0.74 ALDH1A1 (0.47) GPR35MAPTALDH1A1KDM4ECYP3A4
SCHEMBL647033 0.74 MCL1 (0.65) GPR35MAPTALDH1A1KDM4EMEN1
SCHEMBL16396143 0.71 MMP12 (0.47) GPR35ALDH1A1HSD17B10PTPN1POLB
SCHEMBL30340804 0.70 MAPT (0.58) MAPTALDH1A1KDM4ECYP3A4MEN1
SCHEMBL3887754 0.70 MAPT (0.58) MAPTALDH1A1KDM4ECYP3A4MEN1
SCHEMBL16096208 0.69 IKBKB (0.45) MAPTALDH1A1KDM4EMEN1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3004057-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C Research Laboratories (KR) 2016-04-13 EP disclosed
WO-2014196793-A1 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C RESEARCH LABORATORIES (KR) 2014-12-11 WO disclosed