Niacin

Niacin

SCHEMBL1640446

NC(=O)O.O=C(O)c1cccnc1

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.91
APP P05067 1/20 0.91
GAA P10253 1/20 0.91
HCAR3 P49019 1/20 0.91
HCAR2 Q8TDS4 1/20 0.91
F7 P08709 1/20 0.73
F3 P13726 1/20 0.73
SARM1 Q6SZW1 1/20 0.73
SIRT2 Q8IXJ6 1/20 0.73
SIRT6 Q8N6T7 1/20 0.73
SIRT1 Q96EB6 1/20 0.73
SIRT3 Q9NTG7 1/20 0.73
SIRT5 Q9NXA8 1/20 0.73
SIRT4 Q9Y6E7 1/20 0.73
KMO O15229 1/20 0.59
MKNK1 Q9BUB5 2/20 0.58
MKNK2 Q9HBH9 2/20 0.58
PLOD2 O00469 1/20 0.58
HDAC1 Q13547 1/20 0.57
HDAC6 Q9UBN7 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Niacin SCHEMBL20482455 0.96 ALDH1A1 (0.91) ALDH1A1APPGAAHCAR3HCAR2
Niacin SCHEMBL30844065 0.96
Niacin SCHEMBL28292236 0.96 ALDH1A1 (1.00) ALDH1A1APPGAAHCAR3HCAR2
Niacin SCHEMBL3081560 0.96 ALDH1A1 (1.00) ALDH1A1APPGAAHCAR3HCAR2
Niacin SCHEMBL1433 0.96
Niacin SCHEMBL29396199 0.96 ALDH1A1 (1.00) ALDH1A1APPGAAHCAR3HCAR2
Niacin SCHEMBL29349574 0.96
Niacin SCHEMBL150011 0.96 ALDH1A1 (1.00) ALDH1A1APPGAAHCAR3HCAR2
Niacin SCHEMBL31314639 0.94 ALDH1A1 (0.81) ALDH1A1APPGAAHCAR3HCAR2
Niacinamide SCHEMBL1462628 0.94 F7 (0.85) ALDH1A1APPGAAHCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110190267-A1 PRODRUGS OF OPIOIDS AND USES THEREOF SHIRE PHARMACEUTICALS, INC. (US) 2011-08-04 US disclosed
US-20110098278-A1 GALANTAMINE AMINO ACID AND PEPTIDE PRODRUGS AND USES THEREOF SHIRE LLC (US) 2011-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110098278-A1 GALANTAMINE AMINO ACID AND PEPTIDE PRODRUGS AND USES THEREOF PEPD, VIP, GALR1 ALDH1A1 3187/4885APP 18/4885GAA 53/4885
US-20110190267-A1 PRODRUGS OF OPIOIDS AND USES THEREOF OPRK1, OPRL1, OPRM1 ALDH1A1 225/4885APP 2892/4885GAA 1081/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.