SCHEMBL16430680

SCHEMBL16430680

CN(C(=O)Cl)C1CCN(C(C)(C)C)CC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.35
ALDH1A1 P00352 2/20 0.33
CCR5 P51681 1/20 0.32
HSD11B1 P28845 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
L3MBTL3 Q96JM7 1/20 0.32
KCNH2 Q12809 1/20 0.32
TSHR P16473 1/20 0.31
NPY5R Q15761 2/20 0.31
ATM Q13315 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10205080 0.83 VNN1 (0.38) PDK2CCR5L3MBTL3
SCHEMBL3934037 0.83 CCR5 (0.35) PDK2ALDH1A1CCR5HRH3L3MBTL3
SCHEMBL17589228 0.81 DPP4 (0.36) PDK2ALDH1A1CCR5HSD11B1L3MBTL3
SCHEMBL17589231 0.81 PDK2 (0.33) PDK2ALDH1A1CCR5L3MBTL3ATM
SCHEMBL10205061 0.80 VNN1 (0.40) PDK2CCR5HSD11B1KCNH2
SCHEMBL27926085 0.80 HSD11B1 (0.34) PDK2ALDH1A1HSD11B1
SCHEMBL17589227 0.79 CCR5 (0.38) PDK2CCR5HSD11B1L3MBTL3NPY5R
SCHEMBL16219518 0.79 PDK2 (0.36) PDK2CCR5L3MBTL3KCNH2
SCHEMBL10205070 0.79 CCR5 (0.39) ALDH1A1CCR5HSD11B1KCNH2DRD2
SCHEMBL16439286 0.79 ALDH1A1 (0.48) ALDH1A1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3027610-A1 UREA COMPOUNDS AND THEIR USE AS FAAH ENZYME INHIBITORS BIAL - Portela & Cª S.A. (PT) 2016-06-08 EP disclosed
WO-2015016728-A1 UREA COMPOUNDS AND THEIR USE AS FAAH ENZYME INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2015-02-05 WO disclosed
WO-2015016729-A1 UREA COMPOUNDS AND THEIR USE AS FAAH ENZYME INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2015-02-05 WO disclosed