SCHEMBL1644169

SCHEMBL1644169

CCOC(=O)C(=O)c1cccc(OC)c1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.51
MAPT P10636 3/20 0.51
MEN1 O00255 3/20 0.51
LMNA P02545 2/20 0.51
PLIN1 O60240 1/20 0.51
POLB P06746 1/20 0.51
PLIN5 Q00G26 1/20 0.51
ABHD5 Q8WTS1 1/20 0.51
GAA P10253 1/20 0.46
NPSR1 Q6W5P4 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KAT6A Q92794 1/20 0.44
TSHR P16473 2/20 0.42
PKM P14618 1/20 0.42
CYP19A1 P11511 1/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29665865 1.00 KMT2A (0.51) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL27585725 0.84 TSHR (0.58) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL28927886 0.84 KMT2A (0.51) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL28766154 0.84 KMT2A (0.51) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL4589656 0.84 KMT2A (0.60) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL30322741 0.84 KMT2A (0.60) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL4590566 0.83 LMNA (0.52) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL29636596 0.82 LMNA (0.46) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL29362469 0.82 LMNA (0.46) KMT2AMAPTMEN1LMNAPLIN1
SCHEMBL1643613 0.82 LMNA (0.46) KMT2AMAPTMEN1LMNAPLIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109666001-B Method for preparing Elagolix intermediate by multi-step method 安徽华胜医药科技有限公司 2022-06-17 CN claimed
US-11459305-B2 Processes for the preparation of uracil derivatives NEUROCRINE BIOSCIENCES, INC. (US) 2022-10-04 US disclosed
CN-109666001-B Method for preparing Elagolix intermediate by multi-step method 安徽华胜医药科技有限公司 2022-06-17 CN disclosed
US-11339131-B2 Process for preparing elagolix sodium and intermediates thereof SCINOPHARM TAIWAN, LTD. (TW) 2022-05-24 US disclosed
US-20210078956-A1 PROCESS FOR PREPARING ELAGOLIX SODIUM AND INTERMEDIATES THEREOF SCINOPHARM TAIWAN, LTD. (TW) 2021-03-18 US disclosed
US-20200255387-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. 2020-08-13 US disclosed
US-20200255387-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. 2020-08-13 US disclosed
US-20190321363-A1 PROCESS FOR THE PREPARATION OF ELAGOLIX SODIUM AND ITS POLYMORPH DR. REDDY'S LABORATORIES LIMITED (IN) 2019-10-24 US disclosed
US-20190218191-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. 2019-07-18 US disclosed
US-20190218191-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. 2019-07-18 US disclosed
US-9382214-B2 Processes for the preparation of uracil derivatives Neurocine Biosciences, Inc. (US) 2016-07-05 US disclosed
US-9382214-B2 Processes for the preparation of uracil derivatives Neurocine Biosciences, Inc. (US) 2016-07-05 US disclosed
US-8765948-B2 Processes for the preparation of uracil derivatives NEUROCRINE BIOSCIENCES, INC. (US) 2014-07-01 US disclosed
US-8765948-B2 Processes for the preparation of uracil derivatives NEUROCRINE BIOSCIENCES, INC. (US) 2014-07-01 US disclosed
US-8765948-B2 Processes for the preparation of uracil derivatives NEUROCRINE BIOSCIENCES, INC. (US) 2014-07-01 US disclosed
US-20110098472-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. 2011-04-28 US disclosed
US-20110098472-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. 2011-04-28 US disclosed
US-20110098472-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. 2011-04-28 US disclosed
WO-2009062087-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. (US) 2009-05-14 WO disclosed
WO-2009062087-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES NEUROCRINE BIOSCIENCES, INC. (US) 2009-05-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200255387-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES GNRHR, FSHR, GHRHR KMT2A 2736/4885MAPT 3982/4885MEN1 1068/4885
US-11339131-B2 Process for preparing elagolix sodium and intermediates thereof OGG1, ELP1, UNG KMT2A 1754/4885MAPT 4291/4885MEN1 2003/4885
US-20190218191-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES GNRHR, FSHR, GHRHR KMT2A 2736/4885MAPT 3982/4885MEN1 1068/4885
US-20110098472-A1 PROCESSES FOR THE PREPARATION OF URACIL DERIVATIVES GNRHR, FSHR, GHRHR KMT2A 2736/4885MAPT 3982/4885MEN1 1068/4885
US-20210078956-A1 PROCESS FOR PREPARING ELAGOLIX SODIUM AND INTERMEDIATES THEREOF OGG1, ELP1, UNG KMT2A 1754/4885MAPT 4291/4885MEN1 2003/4885
US-20190321363-A1 PROCESS FOR THE PREPARATION OF ELAGOLIX SODIUM AND ITS POLYMORPH PHAX, ELP1, DIS3 KMT2A 2412/4885MAPT 812/4885MEN1 3131/4885
US-11459305-B2 Processes for the preparation of uracil derivatives GNRHR, FSHR, GHRHR KMT2A 2736/4885MAPT 3982/4885MEN1 1068/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.