SCHEMBL16447355

SCHEMBL16447355

CC(C)(C)OC(=O)N1CCC(c2ccc(CN)cc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.57
GPR119 Q8TDV5 8/20 0.54
THRB P10828 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MAPT P10636 1/20 0.50
DDB1 Q16531 1/20 0.48
CRBN Q96SW2 1/20 0.48
WNT3A P56704 1/20 0.48
STS P08842 1/20 0.47
PTPN2 P17706 1/20 0.47
PTPN1 P18031 1/20 0.47
PTPN6 P29350 1/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TP53 P04637 1/20 0.47
PDE4B Q07343 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19539597 0.92 PDE4B (0.55) NAMPTGPR119THRBKDM4EMAPT
SCHEMBL22638944 0.90 NAMPT (0.55) NAMPTGPR119THRBKDM4EMAPT
SCHEMBL2252152 0.88 GPR119 (0.60) NAMPTGPR119THRBKDM4EMAPT
SCHEMBL10243179 0.88 NAMPT (0.58) NAMPTGPR119THRBKDM4EMAPT
SCHEMBL1668728 0.88 TPSAB1 (0.54) NAMPTTHRBKDM4EMAPTGAA
SCHEMBL25273106 0.87 NAMPT (0.57) NAMPTGPR119THRBKDM4EMAPT
SCHEMBL5577703 0.87 NAMPT (0.57) NAMPTGPR119THRBKDM4EMAPT
SCHEMBL31420570 0.86 KDM4E (0.46) NAMPTGPR119KDM4EPDE4B
SCHEMBL14790769 0.86 NAMPT (0.56) NAMPTGPR119THRBKDM4EMAPT
SCHEMBL3529237 0.86 NAMPT (0.56) NAMPTGPR119THRBKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4581025-A1 PYRIDAZINON DERIVATIVES AS KAT2 DEGRADERS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS Auron Therapeutics, Inc. (US) 2025-07-09 EP disclosed
WO-2024050078-A1 PYRIDAZINON DERIVATIVES AS KAT2 DEGRADERS FOR THE TREATMENT OF PROLIFERATIVE DISORDERS AURON THERAPEUTICS, INC. (US) 2024-03-07 WO disclosed
EP-4294389-A1 TRPM8 AGONISTS AS COOLING AGENTS AND FOR THE TREATMENT OF DISEASE Concentric Analgesics, Inc. (US) 2023-12-27 EP disclosed
US-20230014173-A1 Antibacterial Compounds JANSSEN SCIENCES IRELAND UC (IE) 2023-01-19 US disclosed
WO-2022178030-A1 TRPM8 AGONISTS AS COOLING AGENTS AND FOR THE TREATMENT OF DISEASE Concentric Analgesics, Inc. (US) 2022-08-25 WO disclosed
US-11180472-B2 Antibacterial compounds JANSSEN SCIENCES IRELAND UC (IE) 2021-11-23 US disclosed
US-20200239434-A1 ANTIBACTERIAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2020-07-30 US disclosed
US-20190330189-A1 ANTIBACTERIAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2019-10-31 US disclosed
US-10364232-B2 Antibacterial compounds JANSSEN SCIENCES IRELAND UC (IE) 2019-07-30 US disclosed
US-20180186768-A1 Antibacterial Compounds JANSSEN SCIENCES IRELAND UC (IE) 2018-07-05 US disclosed
WO-2015014993-A2 ANTI-INFECTIVE COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2015-02-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11180472-B2 Antibacterial compounds FDPS, SQOR, NDUFS3 NAMPT 138/4885GPR119 4679/4885THRB 3481/4885
US-20190330189-A1 ANTIBACTERIAL COMPOUNDS FDPS, SQOR, NDUFS3 NAMPT 138/4885GPR119 4679/4885THRB 3481/4885
US-10364232-B2 Antibacterial compounds FDPS, SQOR, NDUFS3 NAMPT 138/4885GPR119 4679/4885THRB 3481/4885
US-20180186768-A1 Antibacterial Compounds FDPS, SQOR, NDUFS3 NAMPT 138/4885GPR119 4679/4885THRB 3481/4885
US-20230014173-A1 Antibacterial Compounds FDPS, SQOR, NDUFS3 NAMPT 138/4885GPR119 4679/4885THRB 3481/4885
US-20200239434-A1 ANTIBACTERIAL COMPOUNDS FDPS, SQOR, NDUFS3 NAMPT 138/4885GPR119 4679/4885THRB 3481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.