SCHEMBL16655428

SCHEMBL16655428

O=C(O)c1nn(C2CCCCO2)cc1-c1ccnc2[nH]ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 6/20 0.46
AURKA O14965 5/20 0.46
PIK3C3 Q8NEB9 2/20 0.40
CHEK1 O14757 5/20 0.39
PDCD1 Q15116 5/20 0.39
CD274 Q9NZQ7 5/20 0.39
NUDT1 P36639 1/20 0.39
BRAF P15056 1/20 0.39
CIT O14578 2/20 0.38
IKBKB O14920 2/20 0.37
CHUK O15111 2/20 0.37
INCENP Q9NQS7 2/20 0.37
TPX2 Q9ULW0 1/20 0.37
JAK3 P52333 3/20 0.37
IGF1R P08069 2/20 0.37
ROCK1 Q13464 2/20 0.37
JAK2 O60674 2/20 0.37
DAPK3 O43293 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16655160 0.86 NUDT1 (0.46) AURKBAURKACHEK1PDCD1CD274
SCHEMBL16655108 0.83 AURKB (0.42) AURKBAURKAPIK3C3CHEK1PDCD1
SCHEMBL16655277 0.83 AURKB (0.44) AURKBAURKAPIK3C3CHEK1PDCD1
SCHEMBL1647776 0.79 MAPK14 (0.59) AURKBAURKAPIK3C3BRAFINCENP
SCHEMBL1648278 0.77 AURKB (0.48) AURKBAURKAPIK3C3BRAFCIT
SCHEMBL16655062 0.76 AURKB (0.57) AURKBAURKAPIK3C3NUDT1IKBKB
SCHEMBL1646703 0.76 NUDT1 (0.53) AURKBAURKAPIK3C3NUDT1BRAF
SCHEMBL1648143 0.74 BRAF (0.46) AURKBAURKANUDT1BRAFIKBKB
SCHEMBL25173844 0.70 CYP4F2 (0.39) CD274PRKAA1
SCHEMBL5808316 0.70 ALDH1A1 (0.36) CD274RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057972-A1 NOVEL COMPOSITIONS, USES AND METHODS FOR THEIR PREPARATION Jin, V (US) 2016-08-24 EP disclosed
WO-2015057695-A1 NOVEL COMPOSITIONS, USES AND METHODS FOR THEIR PREPARATION JIN BOHAN (US) 2015-04-23 WO disclosed