SCHEMBL1646804

SCHEMBL1646804

COc1cc(CN2CCC(NC(=O)N(Cc3ccccc3)Cc3ccc(C)cc3)CC2)ccc1O

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.61
MCHR1 Q99705 3/20 0.61
KDM4E B2RXH2 2/20 0.58
ALOX15 P16050 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SIGMAR1 Q99720 6/20 0.57
TSHR P16473 1/20 0.56
ALDH1A1 P00352 1/20 0.54
BCHE P06276 1/20 0.52
ACHE P22303 1/20 0.52
CCR8 P51685 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3708052 0.82 MCHR1 (0.70) HRH3MCHR1KDM4ESIGMAR1ALDH1A1
SCHEMBL341816 0.82 ACHE (0.51) MCHR1KDM4EALOX15TDP1SIGMAR1
SCHEMBL6310838 0.79 SIGMAR1 (0.58) HRH3MCHR1SIGMAR1ALDH1A1ACHE
SCHEMBL5540732 0.78 MCHR1 (0.50) HRH3MCHR1TSHRALDH1A1ACHE
SCHEMBL9871141 0.73 MCHR1 (0.76) MCHR1KDM4ESIGMAR1ALDH1A1
SCHEMBL14543174 0.73 SIGMAR1 (0.58) MCHR1KDM4EALOX15TDP1SIGMAR1
SCHEMBL11098754 0.72 GAA (0.59) KDM4ETDP1TSHRALDH1A1BCHE
SCHEMBL10107601 0.71 SLC6A12 (0.83) MCHR1SIGMAR1ACHE
SCHEMBL6500308 0.71 SIGMAR1 (0.81) MCHR1SIGMAR1CCR8
SCHEMBL1789399 0.71 MCHR1 (0.76) MCHR1SIGMAR1TSHRACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4664564-B2 2011-04-06 JP claimed
JP-2003531829-A 2003-10-28 JP claimed
EP-1263729-A1 AZACYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF SEROTONIN RELATED DISEASES Acadia Pharmaceuticals Inc. (US) 2002-12-11 EP claimed
WO-2001066521-A1 AZACYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF SEROTONIN RELATED DISEASES ACADIA PHARMACEUTICALS, INC. (US) 2001-09-13 WO claimed