SCHEMBL16481978

SCHEMBL16481978

Cc1c[nH]c(-c2cccc(Cl)c2C)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.45
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
ALDH1A1 P00352 4/20 0.37
CNR2 P34972 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
AR P10275 1/20 0.35
KDM4E B2RXH2 2/20 0.34
DCUN1D1 Q96GG9 2/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HSD11B1 P28845 2/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3322110 0.86 MGAM (0.47) IDO1MGAMGAASIMGAM2
SCHEMBL21163205 0.84 ADORA2A (0.36) IDO1MGAMGAASIMGAM2
SCHEMBL29565108 0.83 KMO (0.38) IDO1MGAMGAASIMGAM2
SCHEMBL17069012 0.82 NUDT1 (0.36) MGAMGAASIMGAM2ALDH1A1
SCHEMBL4591602 0.80 KDM4E (0.42) MGAMGAASIMGAM2ALDH1A1
SCHEMBL17194967 0.77 NOTUM (0.35) SMN1; SMN2ARHPGD
SCHEMBL21163207 0.77 MEN1 (0.35) GAAALDH1A1NPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL4345831 0.76 HPGD (0.38) MGAMGAASIMGAM2ALDH1A1
SCHEMBL21091021 0.74 ADRA2A (0.31) SMN1; SMN2HPGD
SCHEMBL24360032 0.74 DCUN1D1 (0.50) IDO1GAAALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014057435-A1 OREXIN RECEPTOR ANTAGONISTS WHICH ARE [ORTHO BI (HETERO )ARYL]-[2-(META BI (HETERO )ARYL)-PYRROLIDIN-1-YL]-METHANONE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2014-04-17 WO disclosed