SCHEMBL21163205

SCHEMBL21163205

Cc1c[nH]c(-c2ccccc2Cc2c[nH]c(-c3cccc(Cl)c3C)n2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
IDO1 P14902 1/20 0.35
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.32
LMNA P02545 2/20 0.31
HPGD P15428 1/20 0.31
ALOX12 P18054 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RAB9A P51151 1/20 0.30
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30
FABP4 P15090 2/20 0.30
FABP3 P05413 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16481978 0.84 IDO1 (0.45) IDO1MGAMGAASIMGAM2
SCHEMBL3322110 0.75 MGAM (0.47) IDO1MGAMGAASIMGAM2
SCHEMBL21163207 0.73 MEN1 (0.35) GAASMN1; SMN2LMNAHPGDNPC1
SCHEMBL29565108 0.70 KMO (0.38) IDO1MGAMGAASIMGAM2
SCHEMBL17069012 0.69 NUDT1 (0.36) MGAMGAASIMGAM2SMN1; SMN2
SCHEMBL8973406 0.69 L3MBTL1 (0.40) ADORA2AADORA1SMN1; SMN2LMNAL3MBTL1
SCHEMBL10792280 0.68 SMN1; SMN2 (0.49) ADORA2AADORA1IDO1SMN1; SMN2LMNA
SCHEMBL4591602 0.67 KDM4E (0.42) ADORA2AADORA1MGAMGAASI
Hydrochloric Acid SCHEMBL4345831 0.67 HPGD (0.38) MGAMGAASIMGAM2SMN1; SMN2
SCHEMBL24360032 0.66 DCUN1D1 (0.50) IDO1GAASMN1; SMN2HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906553-B1 OREXIN RECEPTOR ANTAGONISTS WHICH ARE [ORTHO BI (HETERO )ARYL]-[2-(META BI (HETERO)ARYL)-PYRROLIDIN-1-YL]-METHANONE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2019-06-26 EP disclosed