SCHEMBL21163207

SCHEMBL21163207

CCc1cccc(-c2nc(C)c[nH]2)c1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.35
RAB9A P51151 2/20 0.35
KMT2A Q03164 2/20 0.35
GAA P10253 1/20 0.35
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33
HTR1A P08908 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
TRPA1 O75762 1/20 0.33
ELANE P08246 1/20 0.33
CCNT1 O60563 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CDK9 P50750 1/20 0.32
NPC1 O15118 1/20 0.32
ATM Q13315 1/20 0.32
HPGD P15428 2/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17069012 0.80 NUDT1 (0.36) RAB9AGAATRPA1NPC1ATM
SCHEMBL16481978 0.77 IDO1 (0.45) RAB9AKMT2AGAANPC1HPGD
SCHEMBL17194967 0.74 NOTUM (0.35) GABRA1GABRB2TRPA1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL4345831 0.73 HPGD (0.38) MEN1RAB9AKMT2AGAANPC1
SCHEMBL21163205 0.73 ADORA2A (0.36) RAB9AGAANPC1HPGDALDH1A1
SCHEMBL21091021 0.72 ADRA2A (0.31) HPGDCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL24360032 0.72 DCUN1D1 (0.50) MEN1RAB9AKMT2AGAATRPA1
SCHEMBL29724732 0.71 KDM4E (0.48) GAAHPGDKDM4EHSD17B10CYP1A2
SCHEMBL535697 0.71 KDM4E (0.48) GAAHPGDKDM4EHSD17B10CYP1A2
SCHEMBL15527240 0.70 CD44 (0.39) MEN1RAB9AKMT2AGAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906553-B1 OREXIN RECEPTOR ANTAGONISTS WHICH ARE [ORTHO BI (HETERO )ARYL]-[2-(META BI (HETERO)ARYL)-PYRROLIDIN-1-YL]-METHANONE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2019-06-26 EP disclosed