SCHEMBL16498482

SCHEMBL16498482

[O-][n+]1ccc(-c2nc3cc(-c4ccc5[nH]c(-c6ccncc6)nc5c4)ccc3[nH]2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 4/20 0.53
PKN1 Q16512 4/20 0.53
PKN2 Q16513 4/20 0.53
HPGD P15428 3/20 0.52
RHEB Q15382 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
HSD17B10 Q99714 1/20 0.52
NPC1 O15118 3/20 0.48
RAB9A P51151 2/20 0.48
SCD O00767 1/20 0.47
GUSB P08236 1/20 0.46
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ridinilazole SCHEMBL413723 0.88 ALDH1A1 (0.66) ALDH1A1KDM4EPKN1PKN2HPGD
Ridinilazole SCHEMBL29379856 0.88 ALDH1A1 (0.66) ALDH1A1KDM4EPKN1PKN2HPGD
Ridinilazole SCHEMBL17867397 0.82 NPC1 (0.65) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16498509 0.81 KDM4E (0.57) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL22906080 0.79 ALDH1A1 (0.58) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL6263502 0.79 ALDH1A1 (0.58) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL14834116 0.78 KDM4E (0.54) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16499476 0.77 ALDH1A1 (0.65) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL16499516 0.77 ALDH1A1 (0.53) ALDH1A1KDM4EPKN1PKN2HPGD
SCHEMBL19994448 0.77 ALDH1A1 (0.59) ALDH1A1KDM4EPKN1PKN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151620-A1 COMPOUNDS FOR THE TREATMENT OF CLOSTRIDIUM DIFFICILE ASSOCIATED DISEASE SUMMIT CORPORATION PLC (GB) 2011-12-08 WO claimed
WO-2011151620-A1 COMPOUNDS FOR THE TREATMENT OF CLOSTRIDIUM DIFFICILE ASSOCIATED DISEASE SUMMIT CORPORATION PLC (GB) 2011-12-08 WO disclosed