Methylpyrrolidone

Methylpyrrolidone

SCHEMBL165029

CN1CCCC1=O.CN1CCCC1=O.O

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Methylpyrrolidone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD known ✓ O00329 1/20 0.41
MEN1 known ✓ O00255 3/20 0.39
BRD4 O60885 1/20 0.94
BRD2 P25440 1/20 0.94
INMT O95050 2/20 0.46
GAA P10253 4/20 0.39
KMT2A Q03164 4/20 0.39
MAPT P10636 3/20 0.39
ALDH1A1 P00352 3/20 0.39
PSMD14 O00487 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 3/20 0.38
KDM4E B2RXH2 1/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
CASP1 P29466 1/20 0.37
HSD17B10 Q99714 1/20 0.37
USP2 O75604 1/20 0.36
IDE P14735 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylpyrrolidone SCHEMBL392259 1.00
Methylpyrrolidone SCHEMBL28609570 0.97
Methylpyrrolidone SCHEMBL29239623 0.97
Methylpyrrolidone SCHEMBL10656247 0.97 BRD4 (0.90) BRD4BRD2INMTPIK3CDGAA
Methylpyrrolidone SCHEMBL28300602 0.97
Methylpyrrolidone SCHEMBL8055062 0.97 BRD4 (1.00) BRD4BRD2INMTPIK3CDGAA
Methylpyrrolidone SCHEMBL5423326 0.97
Methylpyrrolidone SCHEMBL487 0.97
Methylpyrrolidone SCHEMBL1255511 0.97 BRD4 (1.00) BRD4BRD2INMTPIK3CDGAA
Methylpyrrolidone SCHEMBL31164528 0.95 BRD4 (0.85) BRD4BRD2INMTPIK3CDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024080370-A1 PILLARARENE COMPLEX ダイキン工業株式会社 2024-04-18 WO disclosed
WO-2024080369-A1 PILLARARENE COMPLEX ダイキン工業株式会社 2024-04-18 WO disclosed
WO-2024080376-A1 PILLARARENE COMPLEX ダイキン工業株式会社 2024-04-18 WO disclosed
EP-4291588-A1 REDUCTION OF MONOMERIC ISOCYANATES BY POROUS MATERIAL BASF SE (DE) 2023-12-20 EP disclosed
CN-116829611-A Reduction of monomeric isocyanates by porous materials 巴斯夫欧洲公司 2023-09-29 CN disclosed
WO-2023157982-A1 ISOLATION METHOD ダイキン工業株式会社 2023-08-24 WO disclosed
CN-111936667-B Method for producing laminate 大金工业株式会社 2022-12-13 CN disclosed
US-10888838-B2 Porous films comprising metal-organic framework materials BASF SE (DE) 2021-01-12 US disclosed
CN-111936667-A Method for producing laminate 大金工业株式会社 2020-11-13 CN disclosed
EP-3311913-B1 POROUS FILMS COMPRISING METAL-ORGANIC FRAMEWORK MATERIALS BASF SE (DE) 2020-05-06 EP disclosed
US-20120049110-A1 Process For Producing A Carbon-Comprising Composite BASF SE (DE) 2012-03-01 US disclosed
US-20120016066-A1 Biodegradable Material Composed Of A Polymer Comprising A Porous Metal-Organic Framework BASF SE (DE) 2012-01-19 US disclosed
US-20110265654-A1 VACUUM INSULATION UNITS COMPRISING GETTER MATERIALS BASF SE (DE) 2011-11-03 US disclosed
US-20100133280-A1 GAS PRESSURE VESSEL COMPRISING A MIXTURE COMPRISING A METAL ORGANIC FRAMEWORK AND ALSO A LATENT HEAT STORE BASF SE (DE) 2010-06-03 US disclosed
US-20100126344-A1 MIXTURE COMPRISING A METAL ORGANIC FRAMEWORK AND ALSO A LATENT HEAT STORE BASF SE (DE) 2010-05-27 US disclosed
US-20090312591-A1 METHOD FOR PRODUCING PROPENE FROM PROPANE BASF SE (DE) 2009-12-17 US disclosed
US-7534303-B2 Liquid absorption by metal-organic frameworks BASF AKTIENGESELLSCHAFT (DE) 2009-05-19 US disclosed
US-20060210458-A1 bringing the liquid into contact with at least one sorbent comprising a porous metal-organic framework, the framework taking up the liquid and comprising at least one at least bidentate organic compound having a coordinate bond to at least one metal ion BASF AKTIENGESELLSCHAFT (DE) 2006-09-21 US disclosed
EP-0703934-A1 PROCESS FOR PRODUCING DECORATIVE MULTIPLE-LAYER VARNISH COATINGS Herberts Gesellschaft mit beschränkter Haftung (DE) 1996-04-03 EP disclosed
WO-1995028428-A1 PROCESS FOR PRODUCING DECORATIVE MULTIPLE-LAYER VARNISH COATINGS Herberts Gesellschaft mit beschränkter Haftung (DE) 1995-10-26 WO disclosed