SCHEMBL165074

SCHEMBL165074

N#Cc1cc(Cl)cc(Cl)c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.41
CYP3A4 P08684 5/20 0.39
ALDH1A1 P00352 4/20 0.39
TRPV4 Q9HBA0 1/20 0.38
KHK P50053 1/20 0.37
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
CLK4 Q9HAZ1 2/20 0.35
CSNK1A1 P48729 1/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 2/20 0.34
XDH P47989 1/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29421236 1.00 GPR35 (0.41) GPR35CYP3A4ALDH1A1TRPV4KHK
SCHEMBL9477728 0.88 KHK (0.41) GPR35CYP3A4ALDH1A1TRPV4KHK
SCHEMBL2435542 0.82 CYP3A4 (0.56) CYP3A4ALDH1A1TRPV4KHKKDM4E
SCHEMBL11028824 0.80 CYP3A4 (0.37) CYP3A4ALDH1A1TRPV4KHKKDM4E
SCHEMBL793224 0.78 KHK (0.43) CYP3A4ALDH1A1TRPV4KHKKDM4E
SCHEMBL5331538 0.78 XDH (0.40) CYP3A4ALDH1A1TRPV4KHKKDM4E
SCHEMBL6119734 0.78 CYP3A4 (0.36) GPR35CYP3A4ALDH1A1TRPV4KHK
SCHEMBL11040450 0.78 ADRB2 (0.41) CYP3A4KHKKDM4EMEN1CYP1A2
SCHEMBL22120138 0.78 KHK (0.47) GPR35CYP3A4ALDH1A1TRPV4KHK
SCHEMBL12225147 0.78 ALDH1A1 (0.36) CYP3A4ALDH1A1KHKKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114149409-B (hetero) aryl amide compound with protein kinase inhibition activity 中国药科大学 2024-03-22 CN disclosed
CN-115551848-A Heterocyclic compounds for controlling invertebrate pests 巴斯夫欧洲公司 2022-12-30 CN disclosed
CN-114149409-A (hetero) aryl amide compound with protein kinase inhibitory activity 中国药科大学 2022-03-08 CN disclosed
EP-3705477-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2020-09-09 EP disclosed
US-10662192-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2020-05-26 US disclosed
EP-3216787-B1 INTERMEDIATES FOR THE PREPARATION OF MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2020-02-19 EP disclosed
US-20190144450-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-05-16 US disclosed
US-10240084-B2 Non-crystallizable pi-conjugated molecular glass mixtures, charge transporting molecular glass mixtures, luminescent molecular glass mixtures, or combinations thereof for organic light emitting diodes and other organic electronics and photonics applications MOLECULAR GLASSES, INC. (US) 2019-03-26 US disclosed
EP-3216787-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2017-09-13 EP disclosed
EP-2502911-B1 Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2017-04-05 EP disclosed
EP-0083009-A1 Dispersion dyestuffs BASF Aktiengesellschaft (DE) 1983-07-06 EP disclosed
EP-0062200-A1 Disazo dyestuffs BASF Aktiengesellschaft (DE) 1982-10-13 EP disclosed
EP-0037465-A2 Amino azo compounds BASF Aktiengesellschaft (DE) 1981-10-14 EP disclosed
US-4152114-A POLYESTERS CIBA-GEIGY AG (CH) 1979-05-01 US disclosed
US-4145341-A WATER-SOLUBLE AZO DYES CONTAINING DIAMINOPYRIMIDINE COUPLER COMPONENTS BASF AKTIENGESELLSCHAFT (DE) 1979-03-20 US disclosed
US-4099909-A POLYESTERS CIBA-GEIGY AG (CH) 1978-07-11 US disclosed
US-4016152-A SUITABLE FOR DYEING POLYESTERS BASF AKTIENGESELLSCHAFT (DT) 1977-04-05 US disclosed
US-3974123-A Dyes for thermoplastics BASF AKTIENGESELLSCHAFT (DT) 1976-08-10 US disclosed
US-3963431-A POLYESTER CIBA-GEIGY AG (CH) 1976-06-15 US disclosed
US-3950321-A POLYESTERS BASF AKTIENGESELLSCHAFT (DT) 1976-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190144450-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS CFTR, ABCB1, ABCC2 GPR35 1346/4885CYP3A4 1862/4885ALDH1A1 2165/4885
US-10662192-B2 Modulators of ATP-binding cassette transporters CFTR, ABCB1, ABCC2 GPR35 1346/4885CYP3A4 1862/4885ALDH1A1 2165/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.