SCHEMBL165154

SCHEMBL165154

Cc1ccc(C2CCCN2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.55
CHRM2 P08172 5/20 0.50
CHRM5 P08912 5/20 0.50
CHRM3 P20309 5/20 0.50
CHRM4 P08173 4/20 0.50
CHRM1 P11229 4/20 0.50
CHRNB2 P17787 2/20 0.50
CHRNA7 P36544 2/20 0.50
CHRNA4 P43681 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
CYP2D6 P10635 3/20 0.44
CYP2C19 P33261 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP2A6 P11509 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6179719 1.00 MKNK1 (0.55) MKNK1CHRM2CHRM5CHRM3CHRM4
SCHEMBL7992297 1.00 MKNK1 (0.55) MKNK1CHRM2CHRM5CHRM3CHRM4
SCHEMBL3717223 0.94 MEN1 (0.51) MKNK1CHRM2CHRM5CHRM3CHRM4
SCHEMBL8541954 0.92 MEN1 (0.50) MKNK1CHRM2CHRM5CHRM3CHRM4
SCHEMBL7672102 0.92 MEN1 (0.50) MKNK1CHRM2CHRM5CHRM3CHRM4
SCHEMBL11510901 0.89 MKNK1 (0.48) MKNK1CHRM2CHRM5CHRM3CHRM4
SCHEMBL25625502 0.85 MAPT (0.48) MKNK1CHRNB2CHRNA4CYP2D6MEN1
SCHEMBL24775559 0.81 CHRNB2 (0.52) MKNK1CHRM2CHRM5CHRM3CHRM4
SCHEMBL21507863 0.80 MEN1 (0.42) MKNK1CHRNB2CHRNA4CYP2D6MEN1
SCHEMBL6557404 0.79 CHRNB2 (0.50) MKNK1CHRM2CHRM5CHRM3CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110922098-B Regenerated asphalt mixture and preparation method thereof Honghui building materials Co.,Ltd. (CN) 2021-08-31 CN claimed
CN-110922098-A Regenerated asphalt mixture and preparation method thereof 宏辉建材有限公司 2020-03-27 CN claimed
CN-101945876-B Nitrogen-containing bicyclic compounds active on chronic pain conditions NEUROTUNE AG 2014-04-30 CN claimed
CN-101945876-A Nitrogen-containing bicyclic compounds active on chronic pain conditions NEUROTUNE AG 2011-01-12 CN claimed
CN-119798161-A Preparation method of plant growth regulating substance and multiple uses thereof 贵州工业职业技术学院 2025-04-11 CN disclosed
EP-3715342-B1 FLUOROSULFONYL-CONTAINING COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF ZHONGHONGXIN INVEST HOLDINGS SHENZHEN CO LTD (CN) 2024-08-07 EP disclosed
US-20230331707-A1 PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2023-10-19 US disclosed
EP-4215532-A1 PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2023-07-26 EP disclosed
US-20230192613-A1 Charged Ion Channel Blockers and Methods for Use NOCION THERAPEUTICS INC (US) 2023-06-22 US disclosed
EP-3177611-B1 OPTIONALLY FUSED HETEROCYCLYL-SUBSTITUTED DERIVATIVES OF PYRIMIDINE USEFUL FOR THE TREATMENT OF INFLAMMATORY, METABOLIC, ONCOLOGIC AND AUTOIMMUNE DISEASES NUEVOLUTION AS (DK) 2021-10-06 EP disclosed
EP-3177611-B1 OPTIONALLY FUSED HETEROCYCLYL-SUBSTITUTED DERIVATIVES OF PYRIMIDINE USEFUL FOR THE TREATMENT OF INFLAMMATORY, METABOLIC, ONCOLOGIC AND AUTOIMMUNE DISEASES NUEVOLUTION AS (DK) 2021-10-06 EP disclosed
CN-110922098-B Regenerated asphalt mixture and preparation method thereof Honghui building materials Co.,Ltd. (CN) 2021-08-31 CN disclosed
CN-101945876-A Nitrogen-containing bicyclic compounds active on chronic pain conditions NEUROTUNE AG 2011-01-12 CN disclosed
US-20100135999-A1 QUINOLINE-CARBOXAMIDE DERIVATIVES AS P2Y12 ANTAGONISTS SANOFI-AVENTIS (FR) 2010-06-03 US disclosed
EP-2148871-A1 QUINOLINE-CARBOXAMIDE DERIVATIVES AS P2Y12 ANTAGONISTS Sanofi-Aventis (FR) 2010-02-03 EP disclosed
WO-2008128647-A1 QUINOLINE-CARBOXAMIDE DERIVATIVES AS P2Y12 ANTAGONISTS SANOFI-AVENTIS (FR) 2008-10-30 WO disclosed
EP-1165510-B1 1-ARENESULFONYL-2-ARYL-PYRROLIDINE AND PIPERIDINE DERIVATIVES FOR THE TREATMENT OF CNS DISORDERS HOFFMANN LA ROCHE (CH) 2005-09-28 EP disclosed
EP-1165510-A1 1-ARENESULFONYL-2-ARYL-PYRROLIDINE AND PIPERIDINE DERIVATIVES FOR THE TREATMENT OF CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-02 EP disclosed
US-6284785-B1 HAVING ACTIVITY AS LIGANDS OF METABOTROPIC GLUTAMATE RECEPTORS HOFFMANN- LA ROCHE INC. 2001-09-04 US disclosed
WO-2000058285-A1 1-ARENESULFONYL-2-ARYL-PYRROLIDINE AND PIPERIDINE DERIVATIVES FOR THE TREATMENT OF CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2000-10-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230331707-A1 PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF RIPK1, RIPK4, RIPK3 MKNK1 416/4885CHRM2 4881/4885CHRM5 4883/4885
US-20100135999-A1 QUINOLINE-CARBOXAMIDE DERIVATIVES AS P2Y12 ANTAGONISTS P2RY12, P2RY1, P2RY2 MKNK1 3409/4885CHRM2 38/4885CHRM5 54/4885
US-20230192613-A1 Charged Ion Channel Blockers and Methods for Use TRPV1, TRPV2, TRPV5 MKNK1 3835/4885CHRM2 384/4885CHRM5 306/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.