SCHEMBL165542

SCHEMBL165542

CC(C)c1cc(Cc2cc(C(C)C)c(N)c(C(C)C)c2Cl)cc(C(C)C)c1N

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.40
P2RX3 P56373 1/20 0.31
P2RX2 Q9UBL9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL169186 0.92 P2RX3 (0.34) DHFRP2RX3P2RX2
SCHEMBL166973 0.85 DHFR (0.37) DHFR
SCHEMBL167931 0.84 P2RX3 (0.31) P2RX3P2RX2
SCHEMBL7555970 0.79 DHFR (0.41) DHFRP2RX3P2RX2
SCHEMBL166081 0.77 DHFR (0.35) DHFR
SCHEMBL101727 0.76 DHFR (0.41) DHFRP2RX3P2RX2
SCHEMBL166574 0.76 ALDH1A1 (0.39)
Hydrochloric Acid SCHEMBL15287283 0.74 DHFR (0.40) DHFRP2RX3P2RX2
SCHEMBL165193 0.74 ALDH1A1 (0.36) P2RX3P2RX2
SCHEMBL166582 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638088-A1 HALOGENATION OF 4,4'-METHYLENE-BIS-ANILINES Lonza Ltd (CH) 2013-09-18 EP disclosed
WO-2012028323-A1 HALOGENATION OF 4,4'-METHYLENE-BIS-ANILINES LONZA LTD (CH) 2012-03-08 WO disclosed