SCHEMBL166973

SCHEMBL166973

Cc1cc(Cc2cc(C)c(N)c(C(C)C)c2Cl)cc(C(C)C)c1N

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.37
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
ALOX15 P16050 1/20 0.32
CASP7 P55210 1/20 0.32
HIF1A Q16665 1/20 0.32
HSD17B10 Q99714 1/20 0.32
LDHA P00338 1/20 0.30
LDHB P07195 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL166574 0.88 ALDH1A1 (0.39) ALDH1A1CYP1A2ALOX15CASP7HIF1A
SCHEMBL165542 0.85 DHFR (0.40) DHFR
SCHEMBL166081 0.84 DHFR (0.35) DHFRALDH1A1
SCHEMBL10053903 0.81 THRB (0.32) DHFRALDH1A1
SCHEMBL169186 0.80 P2RX3 (0.34) DHFR
SCHEMBL29893261 0.79 DHFR (0.37) DHFRALDH1A1CYP1A2ALOX15CASP7
SCHEMBL15488 0.79 DHFR (0.37) DHFRALDH1A1CYP1A2ALOX15CASP7
SCHEMBL3870609 0.78 DHFR (0.36) DHFRALDH1A1CYP1A2ALOX15CASP7
SCHEMBL2941908 0.74 ALDH1A1 (0.39) DHFRALDH1A1CYP1A2ALOX15CASP7
SCHEMBL10341214 0.74 ALDH1A1 (0.36) ALDH1A1CYP1A2ALOX15CASP7HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638088-A1 HALOGENATION OF 4,4'-METHYLENE-BIS-ANILINES Lonza Ltd (CH) 2013-09-18 EP disclosed
WO-2012028323-A1 HALOGENATION OF 4,4'-METHYLENE-BIS-ANILINES LONZA LTD (CH) 2012-03-08 WO disclosed