SCHEMBL1660026

SCHEMBL1660026

C=CC1=C(c2cccc(C3(N[S+]([O-])C(C)(C)C)COC3)c2)C(O)OC=C1Oc1ccc(C(F)(F)F)cc1

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 2/20 0.31
BRAF P15056 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6903826 0.72 TGFBR1 (0.31) RAF1BRAF
SCHEMBL23648676 0.70 LMNA (0.41) RAF1BRAF
SCHEMBL6903571 0.64 TGFBR1 (0.30)
SCHEMBL25365005 0.63 MMP13 (0.34) RAF1
SCHEMBL29523581 0.63 MMP13 (0.34) RAF1
SCHEMBL17869557 0.62 SLC6A3 (0.35)
SCHEMBL30212887 0.62 CHRNA1 (0.35)
SCHEMBL28871226 0.61 BRD4 (0.31)
SCHEMBL9919833 0.61 OPRM1 (0.35)
SCHEMBL25355763 0.60 LMNA (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488031-A1 DIARYL ETHER DERIVATIVES AS NOTCH SPARING GAMMA SECRETASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-08-22 EP disclosed
WO-2011046774-A1 DIARYL ETHER DERIVATIVES AS NOTCH SPARING GAMMA SECRETASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-04-21 WO disclosed