SCHEMBL16601583

SCHEMBL16601583

Cc1ccc2c(c1)S(=O)(=O)C(C)(C)C(=O)N2C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
CNR1 P21554 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
CA12 O43570 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 2/20 0.38
CA7 P43166 2/20 0.38
CA9 Q16790 2/20 0.38
CA1 P00915 1/20 0.38
ALDH1A1 P00352 4/20 0.38
LMNA P02545 4/20 0.38
POLB P06746 3/20 0.38
TSHR P16473 2/20 0.38
KDM4E B2RXH2 3/20 0.36
MEN1 O00255 3/20 0.36
HTT P42858 3/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.35
CRHBP P24387 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13962151 0.82 CASP3 (0.42) PKMCNR1GPR55CA12CA2
SCHEMBL13340958 0.80 NR1H3 (0.39) CA12CA2CA4CA7CA9
SCHEMBL16601584 0.80 ALDH1A1 (0.39) PKMCNR1GPR55CA12CA2
SCHEMBL16601582 0.80 ALDH1A1 (0.38) PKMCA12CA2CA4CA7
SCHEMBL13924055 0.77 CA2 (0.51) PKMCA12CA2CA4CA7
SCHEMBL26513514 0.74 MAOA (0.53) PKMCNR1GPR55CA12CA2
SCHEMBL16285367 0.72 CA2 (0.68) PKMCNR1GPR55CA12CA2
SCHEMBL15653115 0.72 CA12 (0.40) CA12CA2CA4CA7CA9
SCHEMBL5985686 0.71 TP53 (0.39) PKMCNR1GPR55CA12CA2
SCHEMBL5539734 0.70 MEN1 (0.56) PKMCNR1GPR55ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8993585-B2 Cyclic amine substituted pyrimidinediamines as PKC inhibitors RIGEL PHARMACEUTICALS, INC. (US) 2015-03-31 US disclosed